SCHEMBL5763172

SCHEMBL5763172

c1ccc2c(N3CCN(CCCc4ccc5c(c4)CNC5)CC3)nsc2c1

nearest known ligand 0.61

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 4/20 0.60
HTR7 P34969 3/20 0.60
DRD2 P14416 2/20 0.58
HTR2A P28223 2/20 0.58
KCNH2 Q12809 1/20 0.58
HTR6 P50406 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6103732 0.81 HTR1A (0.61) HTR1AHTR7DRD2HTR2AKCNH2
SCHEMBL6219456 0.80 HTR1A (0.53) HTR1AHTR7DRD2HTR2AHTR6
SCHEMBL5767158 0.80 HTR1A (0.55) HTR1AHTR7DRD2HTR2AKCNH2
Water SCHEMBL7416199 0.79 KCNH2 (0.67) HTR1AHTR7DRD2HTR2AKCNH2
SCHEMBL6219541 0.79 HTR2A (0.65) HTR1AHTR7DRD2HTR2AHTR6
SCHEMBL5766860 0.79 HTR1A (0.53) HTR1AHTR7DRD2HTR2AKCNH2
SCHEMBL6401515 0.79 HTR1A (0.56) HTR1AHTR7DRD2HTR2AHTR6
SCHEMBL5764327 0.78 HTR1A (0.67) HTR1AHTR7DRD2HTR2AKCNH2
SCHEMBL1322955 0.78 HTR1A (0.63) HTR1AHTR7DRD2HTR2AKCNH2
SCHEMBL6220391 0.78 HTR1A (0.54) HTR1AHTR7DRD2HTR2AKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1701954-A1 N-SUBSTITUTED PIPERIDINE AND PIPERAZINE DERIVATIVES Warner-Lambert Company LLC (US) 2006-09-20 EP disclosed
WO-2005066165-A1 N-SUBSTITUTED PIPERIDINE AND PIPERAZINE DERIVATIVES WARNER-LAMBERT COMPANY LLC (US) 2005-07-21 WO disclosed