SCHEMBL5764150

SCHEMBL5764150

Cc1ccc([N+](=O)[O-])cc1-c1ccnc(N)c1Cl

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.49
TSHR P16473 2/20 0.49
TDP1 Q9NUW8 7/20 0.46
ALDH1A1 P00352 4/20 0.46
CCNB2 O95067 1/20 0.40
CDK1 P06493 1/20 0.40
CCNB1 P14635 1/20 0.40
CCNA2 P20248 1/20 0.40
CDK2 P24941 1/20 0.40
CCNA1 P78396 1/20 0.40
CCNB3 Q8WWL7 1/20 0.40
MAPT P10636 4/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
POLB P06746 1/20 0.39
HTT P42858 1/20 0.39
HSD17B10 Q99714 1/20 0.38
L3MBTL1 Q9Y468 2/20 0.38
LMNA P02545 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2887065 0.75 ALDH1A1 (0.47) CYP3A4TSHRTDP1ALDH1A1MAPT
SCHEMBL31312390 0.75 ALDH1A1 (0.47) CYP3A4TSHRTDP1ALDH1A1CCNB2
SCHEMBL5764154 0.74 ALDH1A1 (0.46) CYP3A4TSHRTDP1ALDH1A1MAPT
SCHEMBL25983830 0.74 ALDH1A1 (0.46) CYP3A4TSHRTDP1ALDH1A1CCNB2
SCHEMBL28793233 0.73 TDP1 (0.47) TSHRTDP1ALDH1A1MEN1KMT2A
SCHEMBL29716088 0.73 TDP1 (0.47) TSHRTDP1ALDH1A1MEN1KMT2A
SCHEMBL7471914 0.72 TDP1 (0.55) CYP3A4TSHRTDP1ALDH1A1MAPT
SCHEMBL4265596 0.70 ALDH1A1 (0.49) CYP3A4TSHRTDP1ALDH1A1MAPT
SCHEMBL31312282 0.70 DYRK1A (0.47) CYP3A4TSHRTDP1ALDH1A1MAPT
Hydrochloric Acid SCHEMBL6571009 0.70 CYP3A4 (0.60) CYP3A4TSHRTDP1ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1675584-A1 SUBSTITUTED BENZAZOLES AND USE THEREOF AS INHIBITORS OF RAF KINASE CHIRON CORPORATION (US) 2006-07-05 EP disclosed
WO-2005032548-A1 SUBSTITUTED BENZAZOLES AND USE THEREOF AS INHIBITORS OF RAF KINASE CHIRON CORPORATION (US) 2005-04-14 WO disclosed
EP-1499311-A1 SUBSTITUTED BENZAZOLES AND USE THEREOF AS RAF KINASE INHIBITORS Chiron Corporation (US) 2005-01-26 EP disclosed
WO-2003082272-A1 SUBSTITUTED BENZAZOLES AND USE THEREOF AS RAF KINASE INHIBITORS CHIRON CORPORATION (US) 2003-10-09 WO disclosed