SCHEMBL5764679

SCHEMBL5764679

CCn1c(=O)c(-c2c(Cl)cccc2Cl)cc2cnc(SC)nc21

nearest known ligand 0.72

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
FGFR1 P11362 5/20 0.64
EGFR P00533 4/20 0.64
WEE1 P30291 1/20 0.55
SRC P12931 1/20 0.51
FGFR2 P21802 1/20 0.51
FGFR4 P22455 1/20 0.51
FGFR3 P22607 1/20 0.51
BTK Q06187 1/20 0.51
ABL1 P00519 1/20 0.49
PSEN1 P49768 1/20 0.49
PSEN2 P49810 1/20 0.49
APH1B Q8WW43 1/20 0.49
NCSTN Q92542 1/20 0.49
APH1A Q96BI3 1/20 0.49
PSENEN Q9NZ42 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29498163 0.88 RIPK2 (0.54) FGFR1EGFRSRCFGFR2FGFR4
SCHEMBL20564694 0.88 FGFR1 (0.56) FGFR1EGFRWEE1SRCFGFR2
SCHEMBL20564693 0.88 RIPK2 (0.54) FGFR1EGFRSRCFGFR2FGFR4
SCHEMBL29498166 0.88 FGFR1 (0.56) FGFR1EGFRWEE1SRCFGFR2
SCHEMBL5762746 0.86 FGFR1 (0.48) FGFR1EGFRWEE1SRCFGFR2
SCHEMBL20563509 0.86 RIPK2 (0.57) FGFR1EGFRSRCFGFR2FGFR4
SCHEMBL29498221 0.86 RIPK2 (0.57) FGFR1EGFRSRCFGFR2FGFR4
SCHEMBL5761991 0.85 FGFR1 (0.70) FGFR1EGFRWEE1SRCFGFR2
SCHEMBL30618265 0.85 FGFR1 (0.70) FGFR1EGFRWEE1SRCFGFR2
SCHEMBL5763110 0.84 FGFR1 (0.72) FGFR1EGFRWEE1SRCFGFR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0823908-B1 PYRIDO[2,3-d]PYRIMIDINES FOR INHIBITING PROTEIN TYROSINE KINASE MEDIATED CELLULAR PROLIFERATION WARNER LAMBERT CO (US) 2006-11-02 EP disclosed
EP-0823908-A1 PYRIDO 2,3-d]PYRIMIDINES FOR INHIBITING PROTEIN TYROSINE KINASE MEDIATED CELLULAR PROLIFERATION WARNER-LAMBERT COMPANY (US) 1998-02-18 EP disclosed
WO-1996034867-A1 PYRIDO[2,3-d]PYRIMIDINES FOR INHIBITING PROTEIN TYROSINE KINASE MEDIATED CELLULAR PROLIFERATION WARNER-LAMBERT COMPANY (US) 1996-11-07 WO disclosed