SCHEMBL5765819

SCHEMBL5765819

CNC(=O)C1CN(c2cc(F)c(C3(C)CN(C=O)C3)c(F)c2)C(=O)O1

nearest known ligand 0.41

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MAOA P21397 6/20 0.41
GRIN1 Q05586 2/20 0.35
GRIN2B Q13224 2/20 0.35
MAOB P27338 3/20 0.32
CALML3 P27482 2/20 0.32
LMNA P02545 1/20 0.32
PTGS1 P23219 1/20 0.32
SDHA P31040 1/20 0.32
F10 P00742 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3035262 1.00 MAOA (0.41) MAOAGRIN1GRIN2BMAOBCALML3
SCHEMBL3035027 0.89 MAOA (0.53) MAOAMAOBCALML3LMNAPTGS1
SCHEMBL3046255 0.87 MAOA (0.41) MAOAGRIN1GRIN2BMAOBCALML3
SCHEMBL3041381 0.85 MAOA (0.40) MAOAGRIN1GRIN2BMAOBCALML3
SCHEMBL3033115 0.76 MAOA (0.53) MAOAMAOBCALML3LMNAPTGS1
SCHEMBL3041348 0.74 MAOA (0.51) MAOAMAOBCALML3LMNAPTGS1
SCHEMBL5764939 0.74 MAOA (0.51) MAOAMAOBCALML3LMNAPTGS1
SCHEMBL4871651 0.74 MAOA (0.47) MAOAGRIN1GRIN2BMAOBCALML3
SCHEMBL4882399 0.74 MAOA (0.43) MAOAGRIN1GRIN2BMAOBCALML3
SCHEMBL3029181 0.73 MAOA (0.46) MAOACALML3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1478629-B1 N-ARYL-2-OXAZOLIDINONE-5-CARBOXAMIDES AND THEIR DERIVATIVES AND THEIR USE AS ANTIBACTERIALS PHARMACIA & UPJOHN CO LLC (US) 2006-10-11 EP disclosed