SCHEMBL5766844

SCHEMBL5766844

CC(C)(C)OC(=O)NC1CCN(c2cccc3ccc(-n4cnc5cc(C(=O)NCCN6CCOCC6)ccc54)nc23)CC1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.49
MAPK1 P28482 1/20 0.49
HPGD P15428 3/20 0.47
KMT2A Q03164 2/20 0.47
MEN1 O00255 1/20 0.47
GAK O14976 1/20 0.45
RIPK2 O43353 1/20 0.45
ULK1 O75385 1/20 0.45
STK10 O94804 1/20 0.45
PRKD3 O94806 1/20 0.45
MAP4K4 O95819 1/20 0.45
LATS1 O95835 1/20 0.45
PAK4 O96013 1/20 0.45
NTRK1 P04629 1/20 0.45
LCK P06239 1/20 0.45
CDK1 P06493 1/20 0.45
APRT P07741 1/20 0.45
RET P07949 1/20 0.45
PDGFRB P09619 1/20 0.45
PHKG2 P15735 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5765634 0.87 ALDH1A1 (0.55) ALDH1A1MAPK1HPGDKMT2AMEN1
SCHEMBL5765302 0.87 GAK (0.52) HPGDKMT2AMEN1GAKRIPK2
SCHEMBL5764652 0.85 MAP4K4 (0.47) ALDH1A1HPGDGAKRIPK2ULK1
SCHEMBL5767002 0.83 MAP4K4 (0.46) ALDH1A1HPGDGAKRIPK2ULK1
SCHEMBL3840314 0.82 MAP4K4 (0.48) HPGDGAKRIPK2ULK1STK10
SCHEMBL3842680 0.80 IRAK4 (0.52) ALDH1A1HPGDGAKRIPK2ULK1
Morpholine SCHEMBL5764394 0.80 IRAK4 (0.52) GAKRIPK2ULK1STK10PRKD3
SCHEMBL5766850 0.80 MAP4K4 (0.45) GAKRIPK2ULK1STK10PRKD3
SCHEMBL5764136 0.80 CKS1B (0.51) HPGDGAKRIPK2ULK1STK10
SCHEMBL4678752 0.79 MAP4K4 (0.73) HPGDGAKRIPK2ULK1STK10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1235825-B1 NOVEL BENZOIMIDAZOLE DERIVATIVES USEFUL AS ANTIPROLIFERATIVE AGENTS PFIZER PROD INC (US) 2006-01-25 EP disclosed