SCHEMBL5768595

SCHEMBL5768595

CC[C@@H](O)[C@@H]1C[C@H](NCC(C)C)CC[C@@H]1N1CCC(NC(=O)c2cccc(C(F)(F)F)c2)C1=O

nearest known ligand 0.61

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 19/20 0.61
CCR5 P51681 4/20 0.61
KCNH2 Q12809 5/20 0.55
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5770110 1.00 CCR2 (0.61) CCR2CCR5KCNH2MEN1KMT2A
SCHEMBL5769129 0.93 CCR2 (0.63) CCR2CCR5KCNH2MEN1KMT2A
SCHEMBL3733104 0.87 CCR2 (0.78) CCR2CCR5KCNH2
SCHEMBL3734930 0.87 CCR2 (0.78) CCR2CCR5KCNH2
SCHEMBL3734932 0.87 CCR2 (0.78) CCR2CCR5KCNH2
SCHEMBL3733100 0.87 CCR2 (0.78) CCR2CCR5KCNH2
SCHEMBL15310518 0.86 CCR2 (0.60) CCR2CCR5KCNH2MEN1KMT2A
SCHEMBL5820063 0.86 CCR2 (0.60) CCR2CCR5KCNH2MEN1KMT2A
SCHEMBL5767261 0.85 CCR2 (0.77) CCR2CCR5KCNH2
SCHEMBL5767886 0.85 CCR2 (0.61) CCR2CCR5KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1656345-A1 CYCLIC DERIVATIVES AS MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY Bristol-Myers Squibb Company (US) 2006-05-17 EP disclosed
WO-2005021500-A1 CYCLIC DERIVATIVES AS MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY BRISTOL-MYERS SQUIBB COMPANY (US) 2005-03-10 WO disclosed