SCHEMBL5770053

SCHEMBL5770053

CC(C)(C)Nc1nccc(-c2cnc3nc(C(F)(F)F)ccn23)n1

nearest known ligand 0.65

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 16/20 0.65
GABRG2 P18507 16/20 0.65
GABRB3 P28472 16/20 0.65
GABRA3 P34903 14/20 0.65
GABRA5 P31644 3/20 0.42
FLT3 P36888 2/20 0.40
IDH1 O75874 1/20 0.40
IDH2 P48735 1/20 0.40
DYRK1A Q13627 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5770189 0.83 GABRA1 (0.74) GABRA1GABRG2GABRB3GABRA3GABRA5
SCHEMBL5768354 0.79 GABRA1 (1.00) GABRA1GABRG2GABRB3GABRA3GABRA5
SCHEMBL5770436 0.76 GABRA1 (1.00) GABRA1GABRG2GABRB3GABRA3GABRA5
SCHEMBL5767966 0.75 GABRA1 (0.60) GABRA1GABRG2GABRB3GABRA3GABRA5
SCHEMBL5770607 0.74 GABRA1 (0.80) GABRA1GABRG2GABRB3GABRA3GABRA5
SCHEMBL5770368 0.74 GABRA1 (1.00) GABRA1GABRG2GABRB3GABRA3GABRA5
SCHEMBL13965269 0.73 IDH1 (0.53) IDH1IDH2
SCHEMBL5773757 0.73 GABRA1 (0.64) GABRA1GABRG2GABRB3GABRA3GABRA5
SCHEMBL5769413 0.73 GABRA1 (0.57) GABRA1GABRG2GABRB3GABRA3GABRA5
SCHEMBL5768345 0.73 GABRA1 (0.57) GABRA1GABRG2GABRB3GABRA3GABRA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1383768-B1 IMIDAZO-PYRIMIDINE DERIVATIVES AS LIGANDS FOR GABA RECEPTORS MERCK SHARP & DOHME (GB) 2006-09-06 EP disclosed