SCHEMBL5774600

SCHEMBL5774600

CC(C)c1csc(C=Cc2cncc(NC(=O)O)c2)n1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALB P02768 2/20 0.51
AKT1 P31749 5/20 0.38
NTRK1 P04629 1/20 0.36
ROCK2 O75116 2/20 0.34
PIM1 P11309 2/20 0.34
PRKACA P17612 2/20 0.34
GSK3A P49840 2/20 0.34
RPS6KA3 P51812 2/20 0.34
PRKCD Q05655 2/20 0.34
ROCK1 Q13464 2/20 0.34
DYRK1A Q13627 2/20 0.34
CDC42BPA Q5VT25 2/20 0.34
FGFR3 P22607 1/20 0.34
LIMK1 P53667 1/20 0.34
KDM4E B2RXH2 1/20 0.33
MEN1 O00255 1/20 0.33
ALDH1A1 P00352 1/20 0.33
TP53 P04637 1/20 0.33
ADRB1 P08588 1/20 0.33
CYP3A4 P08684 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27588135 0.85 ALB (0.44) ALBAKT1NTRK1ROCK2PIM1
SCHEMBL5779562 0.85 ALB (0.44) ALBAKT1NTRK1ROCK2PIM1
SCHEMBL5774563 0.84 ALB (0.69) ALBKDM4EMEN1ALDH1A1TP53
SCHEMBL5776451 0.82 ALB (0.43) ALBAKT1NTRK1DYRK1AKDM4E
SCHEMBL5777728 0.82 ALB (0.43) ALBAKT1NTRK1CYP1A2CYP2D6
SCHEMBL5780463 0.81 ALB (0.81) ALBAKT1NTRK1ROCK2PIM1
SCHEMBL5780685 0.79 AKT1 (0.38) ALBAKT1ROCK2PIM1PRKACA
SCHEMBL27572318 0.76 ALB (0.39) ALB
SCHEMBL5779199 0.76 ALB (0.39) ALB
SCHEMBL5908387 0.76 ALB (0.50) ALBGSK3AKDM4EMEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1652839-A2 Drug efflux pump inhibitor DAIICHI PHARMACEUTICAL CO., LTD. (JP) 2006-05-03 EP disclosed
EP-1227084-B1 DRUG DISCHARGE PUMP INHIBITORS TRINE PHARMACEUTICALS INC (US) 2005-12-14 EP disclosed
EP-1227084-A1 DRUG DISCHARGE PUMP INHIBITORS Microcide Pharmaceuticals, Inc. (US) 2002-07-31 EP disclosed