SCHEMBL5779562

SCHEMBL5779562

CC(C)c1csc(C=Cc2cncc(NC(=O)OC(C)(C)C)c2)n1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALB P02768 2/20 0.44
NAMPT P43490 1/20 0.35
NTRK1 P04629 1/20 0.34
HDAC3 O15379 3/20 0.33
HDAC1 Q13547 3/20 0.33
HDAC2 Q92769 3/20 0.33
HDAC8 Q9BY41 3/20 0.33
SREBF2 Q12772 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
AKT1 P31749 3/20 0.32
CYP17A1 P05093 1/20 0.32
RAB9A P51151 1/20 0.32
HDAC10 Q969S8 2/20 0.32
ABCB1 P08183 1/20 0.32
LCK P06239 1/20 0.32
ADORA2B P29275 1/20 0.32
ROCK2 O75116 1/20 0.32
PIM1 P11309 1/20 0.32
PRKACA P17612 1/20 0.32
FGFR3 P22607 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27588135 1.00 ALB (0.44) ALBNAMPTNTRK1HDAC3HDAC1
SCHEMBL5775071 0.86 ALB (0.60) ALBHDAC3HDAC1HDAC2HDAC8
SCHEMBL5774600 0.85 ALB (0.51) ALBNTRK1HDAC3HDAC1HDAC2
SCHEMBL5779051 0.82 PSMB8 (0.35) NAMPTHDAC3HDAC1HDAC2HDAC8
SCHEMBL27588101 0.82 PSMB8 (0.35) NAMPTHDAC3HDAC1HDAC2HDAC8
SCHEMBL5908485 0.79 ALB (0.44) ALBSREBF2ROCK2DYRK1A
SCHEMBL5776451 0.75 ALB (0.43) ALBNTRK1AKT1DYRK1A
SCHEMBL5777728 0.75 ALB (0.43) ALBNTRK1AKT1
SCHEMBL5780243 0.74 ALB (0.41) ALBHDAC3HDAC1HDAC2HDAC8
SCHEMBL27569393 0.74 ALB (0.41) ALBHDAC3HDAC1HDAC2HDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1652839-A2 Drug efflux pump inhibitor DAIICHI PHARMACEUTICAL CO., LTD. (JP) 2006-05-03 EP disclosed
EP-1227084-B1 DRUG DISCHARGE PUMP INHIBITORS TRINE PHARMACEUTICALS INC (US) 2005-12-14 EP disclosed
EP-1227084-A1 DRUG DISCHARGE PUMP INHIBITORS Microcide Pharmaceuticals, Inc. (US) 2002-07-31 EP disclosed