SCHEMBL5775071

SCHEMBL5775071

CC(C)c1csc(C=Cc2cccc(NC(=O)OC(C)(C)C)c2)n1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALB P02768 2/20 0.60
HDAC3 O15379 5/20 0.43
HDAC1 Q13547 4/20 0.43
HDAC2 Q92769 4/20 0.43
HDAC8 Q9BY41 3/20 0.43
HDAC6 Q9UBN7 2/20 0.43
KDM4E B2RXH2 1/20 0.43
MEN1 O00255 1/20 0.43
ALDH1A1 P00352 1/20 0.43
TP53 P04637 1/20 0.43
ADRB1 P08588 1/20 0.43
CYP3A4 P08684 1/20 0.43
ADORA3 P0DMS8 1/20 0.43
MAPT P10636 1/20 0.43
HPGD P15428 1/20 0.43
PTGS1 P23219 1/20 0.43
KMT2A Q03164 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
HSD17B10 Q99714 1/20 0.43
HDAC10 Q969S8 3/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27588135 0.86 ALB (0.44) ALBHDAC3HDAC1HDAC2HDAC8
SCHEMBL5779562 0.86 ALB (0.44) ALBHDAC3HDAC1HDAC2HDAC8
SCHEMBL5774563 0.85 ALB (0.69) ALBHDAC3HDAC1HDAC2HDAC8
SCHEMBL5908485 0.83 ALB (0.44) ALBCYP3A4
SCHEMBL5777394 0.82 ALB (0.50) ALBHDAC3HDAC1HDAC6KDM4E
SCHEMBL27569393 0.80 ALB (0.41) ALBHDAC3HDAC1HDAC2HDAC8
SCHEMBL5780243 0.80 ALB (0.41) ALBHDAC3HDAC1HDAC2HDAC8
SCHEMBL5779901 0.80 ALB (0.51) ALBKDM4EMEN1ALDH1A1TP53
SCHEMBL9094380 0.78 KDM4E (0.70) ALBKDM4EMEN1ALDH1A1TP53
SCHEMBL9094397 0.78 KDM4E (0.70) ALBKDM4EMEN1ALDH1A1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1652839-A2 Drug efflux pump inhibitor DAIICHI PHARMACEUTICAL CO., LTD. (JP) 2006-05-03 EP disclosed
EP-1227084-B1 DRUG DISCHARGE PUMP INHIBITORS TRINE PHARMACEUTICALS INC (US) 2005-12-14 EP disclosed
EP-1227084-A1 DRUG DISCHARGE PUMP INHIBITORS Microcide Pharmaceuticals, Inc. (US) 2002-07-31 EP disclosed