SCHEMBL5776008

SCHEMBL5776008

CC(C)c1cc(F)cc2c1c(C(=O)c1ccc(Cl)cc1S(C)(=O)=O)c1n2CC[C]1

nearest known ligand 0.42

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TBXA2R P21731 17/20 0.42
PTGER1 P34995 2/20 0.39
PTGFR P43088 1/20 0.39
PTGER3 P43115 1/20 0.39
PTGER2 P43116 1/20 0.39
PTGDR2 Q9Y5Y4 1/20 0.39
CNR2 P34972 1/20 0.31
GPR183 P32249 1/20 0.31
ALDH1A1 P00352 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5835901 0.78 TBXA2R (0.69) TBXA2RPTGER1PTGFRPTGER3PTGER2
SCHEMBL5798298 0.65 TBXA2R (0.63) TBXA2RPTGER1PTGFRPTGER3PTGER2
SCHEMBL14582545 0.61 TBXA2R (0.65) TBXA2RPTGER1PTGFRPTGER3PTGER2
SCHEMBL15281022 0.60 SLC9A1 (0.49) PTGDR2CNR2ALDH1A1
SCHEMBL8606110 0.59 SMN1; SMN2 (0.51) CNR2ALDH1A1
SCHEMBL5778175 0.59 TBXA2R (0.49) TBXA2RPTGDR2
SCHEMBL8490829 0.59 AVPR2 (0.44) CNR2ALDH1A1
SCHEMBL2126878 0.59 SMN1; SMN2 (0.55) ALDH1A1
SCHEMBL28647649 0.58 HTT (0.42) CNR2
SCHEMBL8491568 0.58 CNR2 (0.39) CNR2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1395590-B1 DIHYDROPYRROLO¬1,2-A|INDOLE AND TETRAHYDROPYRIDO¬1,2-A|INDOLE DERIVATIVES AS PROSTAGLANDIN D2 RECEPTOR ANTAGONISTS MERCK FROSST CANADA INC (CA) 2006-09-27 EP disclosed