SCHEMBL5777130

SCHEMBL5777130

CC(C)Oc1cc(S(C)(=O)=O)c2cc3n(c2c1)CCC3CC(=O)O

nearest known ligand 0.44

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 7/20 0.44
S1PR5 Q9H228 3/20 0.44
TBXA2R P21731 9/20 0.41
S1PR4 O95977 2/20 0.37
CYP2C9 P11712 1/20 0.37
FFAR4 Q5NUL3 2/20 0.37
PDE2A O00408 2/20 0.37
PTGDR Q13258 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5835938 0.85 KDM4E (0.34) S1PR1S1PR5FFAR4PTGDR
SCHEMBL5776224 0.85 TBXA2R (0.42) S1PR1S1PR5TBXA2RS1PR4PDE2A
SCHEMBL5778068 0.83 TBXA2R (0.44) S1PR1S1PR5TBXA2RPDE2APTGDR
SCHEMBL5774565 0.82 TBXA2R (0.57) TBXA2RPDE2APTGDR
SCHEMBL5775903 0.82 TBXA2R (0.57) TBXA2RPDE2APTGDR
SCHEMBL5776803 0.77 HTT (0.34)
SCHEMBL5774771 0.76 TBXA2R (0.56) TBXA2RPDE2APTGDR
SCHEMBL5779554 0.75 S1PR1 (0.43) S1PR1S1PR5TBXA2RS1PR4FFAR4
SCHEMBL5777734 0.74 S1PR1 (0.43) S1PR1S1PR5TBXA2RS1PR4
SCHEMBL5775625 0.74 S1PR1 (0.47) S1PR1S1PR5TBXA2RS1PR4FFAR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1395590-B1 DIHYDROPYRROLO¬1,2-A|INDOLE AND TETRAHYDROPYRIDO¬1,2-A|INDOLE DERIVATIVES AS PROSTAGLANDIN D2 RECEPTOR ANTAGONISTS MERCK FROSST CANADA INC (CA) 2006-09-27 EP disclosed