SCHEMBL5776224

SCHEMBL5776224

CS(=O)(=O)c1cc(OS(=O)(=O)C(F)(F)F)cc2c1cc1n2CCC1CC(=O)O

nearest known ligand 0.42

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
TBXA2R P21731 9/20 0.42
PDE2A O00408 3/20 0.42
PTGDR Q13258 3/20 0.42
S1PR1 P21453 8/20 0.41
S1PR4 O95977 1/20 0.39
S1PR5 Q9H228 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5777734 0.85 S1PR1 (0.43) TBXA2RS1PR1S1PR4S1PR5
SCHEMBL5777130 0.85 S1PR1 (0.44) TBXA2RPDE2APTGDRS1PR1S1PR4
SCHEMBL5775903 0.83 TBXA2R (0.57) TBXA2RPDE2APTGDR
SCHEMBL5774565 0.83 TBXA2R (0.57) TBXA2RPDE2APTGDR
SCHEMBL5778068 0.82 TBXA2R (0.44) TBXA2RPDE2APTGDRS1PR1S1PR5
SCHEMBL5774771 0.77 TBXA2R (0.56) TBXA2RPDE2APTGDR
SCHEMBL5775625 0.73 S1PR1 (0.47) TBXA2RS1PR1S1PR4S1PR5
SCHEMBL5772689 0.72 TBXA2R (0.39) TBXA2RPDE2APTGDR
SCHEMBL5776803 0.72 HTT (0.34)
SCHEMBL5777074 0.70 S1PR1 (0.43) TBXA2RS1PR1S1PR4S1PR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1395590-B1 DIHYDROPYRROLO¬1,2-A|INDOLE AND TETRAHYDROPYRIDO¬1,2-A|INDOLE DERIVATIVES AS PROSTAGLANDIN D2 RECEPTOR ANTAGONISTS MERCK FROSST CANADA INC (CA) 2006-09-27 EP disclosed