SCHEMBL5777875

SCHEMBL5777875

CC(C)(C)OC(=O)ON1CC2CNCC(C1)O2

nearest known ligand 0.42

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 1/20 0.30
CHRNB4 P30926 1/20 0.30
CHRNA3 P32297 1/20 0.30
CHRNA4 P43681 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3397031 0.82 CHRNA4 (0.43) CHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL5537141 0.82 CHRNA4 (0.43) CHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL4584160 0.78 CHRM2 (0.35)
SCHEMBL56234 0.78 NR1H2 (0.46) CHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL29707388 0.78 NR1H2 (0.46) CHRNB2CHRNB4CHRNA3CHRNA4
Hydrochloric Acid SCHEMBL2956489 0.76 NR1H2 (0.45) CHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL14764516 0.74 CHRM2 (0.41)
SCHEMBL8329335 0.74 CHRM2 (0.37)
SCHEMBL8329981 0.74 CHRM2 (0.37)
SCHEMBL5777377 0.71 S1PR5 (0.41)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1525202-B1 NOVEL 2,5-DISUBSTITUTED PYRIMIDINE DERIVATIVES BAYER HEALTHCARE AG (DE) 2006-01-11 EP disclosed
EP-1525202-A1 NOVEL 2,5-DISUBSTITUTED PYRIMIDINE DERIVATIVES Bayer HealthCare AG (DE) 2005-04-27 EP disclosed
WO-2004009589-A1 NOVEL 2,5-DISUBSTITUTED PYRIMIDINE DERIVATIVES BAYER HEALTHCARE AG (DE) 2004-01-29 WO disclosed