SCHEMBL5537141

SCHEMBL5537141

CC(C)(C)OC(=O)ON1C[C@H]2CNC[C@H]2C1

nearest known ligand 0.45

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CHRNA4 P43681 17/20 0.43
CHRNB2 P17787 16/20 0.43
CHRNB4 P30926 16/20 0.43
CHRNA3 P32297 16/20 0.43
CHRNA7 P36544 14/20 0.41
NR1H2 P55055 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3397031 1.00 CHRNA4 (0.43) CHRNA4CHRNB2CHRNB4CHRNA3CHRNA7
SCHEMBL5777875 0.82 CHRNB2 (0.30) CHRNA4CHRNB2CHRNB4CHRNA3
SCHEMBL8329981 0.78 CHRM2 (0.37) NR1H2
SCHEMBL8329335 0.78 CHRM2 (0.37) NR1H2
SCHEMBL14764516 0.78 CHRM2 (0.41) NR1H2
SCHEMBL3647706 0.76 NR1H2 (0.31) NR1H2
SCHEMBL4711086 0.76 NR1H2 (0.31) NR1H2
SCHEMBL4584160 0.75 CHRM2 (0.35) NR1H2
SCHEMBL649983 0.75 CHRNB2 (0.65) CHRNA4CHRNB2CHRNB4CHRNA3CHRNA7
SCHEMBL16053523 0.75 CHRNB2 (0.65) CHRNA4CHRNB2CHRNB4CHRNA3CHRNA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1776372-A1 SUBSTITUTED, BICYCLIC 8-PYRROLIDINOXANTHINES, METHOD FOR THE PRODUCTION THEREOF AND THEIR USE AS MEDICAMENTS Sanofi-Aventis Deutschland GmbH (DE) 2007-04-25 EP disclosed
WO-2006015701-A1 SUBSTITUTED, BICYCLIC 8-PYRROLIDINOXANTHINES, METHOD FOR THE PRODUCTION THEREOF AND THEIR USE AS MEDICAMENTS SANOFI-AVENTIS DEUTSCHLAND GMBH (DE) 2006-02-16 WO disclosed