SCHEMBL5777930

SCHEMBL5777930

CC(CF)(CC(O)C(F)F)c1cc(F)cc2c1OCC2

nearest known ligand 0.42

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
NR3C1 P04150 8/20 0.42
PGR P06401 8/20 0.42
NR3C2 P08235 8/20 0.42
PARP1 P09874 1/20 0.40
PTGS1 P23219 1/20 0.34
PTGS2 P35354 1/20 0.34
RIPK1 Q13546 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5779024 0.85 PTGS1 (0.32) NR3C1PGRNR3C2PTGS1PTGS2
SCHEMBL5777927 0.75 NR3C1 (0.48) NR3C1PGRNR3C2PARP1PTGS1
SCHEMBL14146333 0.74 NR3C1 (0.45) NR3C1PGRNR3C2PARP1PTGS1
SCHEMBL19505262 0.74 PARP1 (0.50) NR3C1PGRNR3C2PARP1PTGS1
SCHEMBL14146329 0.73 NR3C1 (0.44) NR3C1PGRNR3C2PARP1PTGS1
SCHEMBL14189079 0.72 NR3C1 (0.48) NR3C1PGRNR3C2PARP1PTGS1
SCHEMBL3649794 0.71 CHRM3 (0.37) NR3C1PGRNR3C2
SCHEMBL675925 0.71 NR3C1 (0.66) NR3C1PGRNR3C2
SCHEMBL4557422 0.71 NR3C1 (0.59) NR3C1PGRNR3C2
SCHEMBL3658042 0.71 NR3C1 (0.52) NR3C1PGRNR3C2PARP1PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1673088-A1 1,1,1- TRIFLUORO-4-PHENYL-4-METHYL-2-(1H-PYRROLO¬2,3-C|PYRIDIN-2-YLMETHYL)PENTAN-2-OL DERIVATIVES AND RELATED COMPOUNDS AS GLUCOCORTICOID LIGANDS FOR THE TREATMENT OF INFLAMMATORY DISEASES AND DIABETES BOEHRINGER INGELHEIM PHARMACEUTICALS INC. (US) 2006-06-28 EP disclosed
WO-2005030213-A1 1,1,1-TRIFLUORO-4-PHENYL-4-METHYL-2-(1H-PYRROLO BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2005-04-07 WO disclosed