SCHEMBL5778738

SCHEMBL5778738

CCc1nc2c(Cl)nc(Cl)cc2[nH]1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 3/20 0.50
GAA P10253 2/20 0.50
ADORA1 P30542 4/20 0.41
ADORA3 P0DMS8 3/20 0.41
ADORA2A P29274 2/20 0.41
DDAH1 O94760 1/20 0.41
MME P08473 1/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
ALDH1A1 P00352 2/20 0.32
KDM4E B2RXH2 1/20 0.32
PTGES O14684 1/20 0.31
CACNA1H O95180 2/20 0.31
GLA P06280 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
RHEB Q15382 2/20 0.31
CCNE2 O96020 1/20 0.31
CDK4 P11802 1/20 0.31
CCND1 P24385 1/20 0.31
CCNE1 P24864 1/20 0.31
CDK2 P24941 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25802549 0.77 AAK1 (0.38) ALDH1A1CACNA1H
SCHEMBL5778409 0.76 HTT (0.56) HTTADORA3SMN1; SMN2ALDH1A1
SCHEMBL29491150 0.76 HTT (0.56) HTTADORA3SMN1; SMN2ALDH1A1
SCHEMBL3209801 0.70 HTT (0.41) HTTGAAADORA1ADORA3ADORA2A
SCHEMBL4363219 0.69 GAA (0.43) HTTGAAADORA1ADORA3ADORA2A
SCHEMBL10284437 0.69 CACNA1H (0.51) HTTGAAADORA1CACNA1HCACNA1G
SCHEMBL18050722 0.69 AR (0.33) HTT
SCHEMBL29439058 0.68 F10 (0.48) HTTGAAADORA1ADORA3ADORA2A
SCHEMBL1918622 0.68 DDAH1 (0.53) HTTGAAADORA1ADORA3ADORA2A
SCHEMBL27997290 0.68 GAA (0.42) HTTGAAADORA1ADORA3ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1472254-A4 PURINE AND ISOSTERIC ANTIBACTERIAL COMPOUNDS GLSYNTHESIS INC (US) 2006-02-15 EP disclosed
US-6926763-B2 Purine and isosteric antibacterial compounds GLSYNTHESIS, INC. (US) 2005-08-09 US disclosed
EP-1472254-A2 PURINE AND ISOSTERIC ANTIBACTERIAL COMPOUNDS Glsynthesis Inc. (US) 2004-11-03 EP disclosed
WO-2003066586-A2 PURINE AND ISOSTERIC ANTIBACTERIAL COMPOUNDS GLSYNTHESIS INC. (US) 2003-08-14 WO disclosed