SCHEMBL5778769

SCHEMBL5778769

NC(=O)C1CC1c1cccc([N+](=O)[O-])c1

nearest known ligand 0.74

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC9A1 P19634 2/20 0.74
TP53 P04637 2/20 0.54
MAPT P10636 3/20 0.51
MEN1 O00255 1/20 0.51
KMT2A Q03164 1/20 0.51
NPSR1 Q6W5P4 1/20 0.51
TSHR P16473 4/20 0.50
LMNA P02545 2/20 0.48
ALDH1A1 P00352 4/20 0.46
HPGD P15428 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
CES2 O00748 1/20 0.45
CES1 P23141 1/20 0.45
CACNA1F O60840 1/20 0.44
ADORA3 P0DMS8 1/20 0.44
CACNA1D Q01668 1/20 0.44
CACNA1S Q13698 1/20 0.44
CACNA1C Q13936 1/20 0.44
PRSS1 P07477 1/20 0.44
PRSS2 P07478 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31406299 0.90 SLC9A1 (0.64) SLC9A1TP53MAPTMEN1KMT2A
SCHEMBL5774969 0.87 SLC9A1 (0.68) SLC9A1TP53MAPTMEN1KMT2A
SCHEMBL5775091 0.87 SLC9A1 (0.67) SLC9A1TP53MAPTMEN1KMT2A
SCHEMBL6902353 0.87 SLC9A1 (0.67) SLC9A1TP53MAPTMEN1KMT2A
SCHEMBL7002979 0.87 SLC9A1 (0.67) SLC9A1TP53MAPTMEN1KMT2A
SCHEMBL29640120 0.85 SLC9A1 (0.65) SLC9A1TP53MAPTMEN1KMT2A
SCHEMBL21200122 0.85 SLC9A1 (0.65) SLC9A1TP53MAPTMEN1KMT2A
SCHEMBL21200120 0.85 SLC9A1 (0.65) SLC9A1TP53MAPTMEN1KMT2A
SCHEMBL30879548 0.82 SLC9A1 (0.62) SLC9A1TP53MAPTMEN1KMT2A
SCHEMBL30879550 0.82 SLC9A1 (0.62) SLC9A1TP53MAPTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1652839-A2 Drug efflux pump inhibitor DAIICHI PHARMACEUTICAL CO., LTD. (JP) 2006-05-03 EP disclosed
EP-1227084-B1 DRUG DISCHARGE PUMP INHIBITORS TRINE PHARMACEUTICALS INC (US) 2005-12-14 EP disclosed
CN-1414951-A Drug discharge pump inhibitor FUNDAMENTAL THERAPEUTICAL INC (US) 2003-04-30 CN disclosed
EP-1227084-A1 DRUG DISCHARGE PUMP INHIBITORS Microcide Pharmaceuticals, Inc. (US) 2002-07-31 EP disclosed