SCHEMBL5778978

SCHEMBL5778978

CC(C)c1csc(C=Cc2cccc(NC(=O)[C@@H]3CCCC[C@@H]3C(=O)O)c2)n1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALB P02768 1/20 0.58
GRK2 P25098 1/20 0.48
CASP6 P55212 1/20 0.48
CASP8 Q14790 1/20 0.48
CTDSP1 Q9GZU7 1/20 0.48
TDP1 Q9NUW8 1/20 0.48
L3MBTL1 Q9Y468 1/20 0.48
APEX1 P27695 1/20 0.48
ALDH1A1 P00352 5/20 0.47
KDM4E B2RXH2 3/20 0.47
MAPT P10636 2/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
TP53 P04637 2/20 0.47
KMT2A Q03164 2/20 0.47
MEN1 O00255 1/20 0.47
ADRB1 P08588 1/20 0.47
CYP3A4 P08684 1/20 0.47
ADORA3 P0DMS8 1/20 0.47
HPGD P15428 1/20 0.47
PTGS1 P23219 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5777169 1.00 ALB (0.58) ALBGRK2CASP6CASP8CTDSP1
SCHEMBL5778584 0.91 ALB (0.60) ALBGRK2CASP6CASP8CTDSP1
SCHEMBL5774563 0.83 ALB (0.69) ALBALDH1A1KDM4EMAPTSMN1; SMN2
SCHEMBL5776470 0.81 ALB (0.57) ALBALDH1A1KDM4EMAPTSMN1; SMN2
SCHEMBL9518151 0.77 GRK2 (0.50) GRK2CASP6CASP8CTDSP1TDP1
SCHEMBL9518146 0.77 GRK2 (0.50) GRK2CASP6CASP8CTDSP1TDP1
SCHEMBL9518140 0.77 GRK2 (0.50) GRK2CASP6CASP8CTDSP1TDP1
SCHEMBL9264563 0.77 ALB (0.71) ALBL3MBTL1ALDH1A1KDM4EMAPT
SCHEMBL9264552 0.77 ALB (0.71) ALBL3MBTL1ALDH1A1KDM4EMAPT
SCHEMBL5775071 0.76 ALB (0.60) ALBALDH1A1KDM4EMAPTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1652839-A2 Drug efflux pump inhibitor DAIICHI PHARMACEUTICAL CO., LTD. (JP) 2006-05-03 EP disclosed
EP-1227084-A1 DRUG DISCHARGE PUMP INHIBITORS Microcide Pharmaceuticals, Inc. (US) 2002-07-31 EP disclosed