SCHEMBL5779214

SCHEMBL5779214

CCCCOC(=O)NC(CNC(=O)c1cn(CCc2ccccc2)c2cc(CNC3N=CCCN3)ccc2c1=O)C(=O)O

nearest known ligand 0.41

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 13/20 0.41
CNR1 P21554 11/20 0.41
ITGB3 P05106 3/20 0.36
ITGAV P06756 3/20 0.36
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34
HPGD P15428 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5782259 0.92 ITGB3 (0.41) CNR2CNR1ITGB3ITGAV
SCHEMBL5778299 0.89 CNR2 (0.45) CNR2CNR1KDM4EALDH1A1HPGD
SCHEMBL5780511 0.87 CNR2 (0.42) CNR2CNR1ITGB3ITGAVALDH1A1
SCHEMBL1072330 0.87 KDM4E (0.35) CNR2ITGB3ITGAVKDM4EALDH1A1
SCHEMBL5779660 0.85 ITGB3 (0.42) ITGB3ITGAV
SCHEMBL5781660 0.84 ITGB3 (0.43) CNR2CNR1ITGB3ITGAVALDH1A1
SCHEMBL5783014 0.83 ITGB3 (0.49) CNR2CNR1ITGB3ITGAV
SCHEMBL5779767 0.82 ITGAV (0.53) ITGB3ITGAV
SCHEMBL5780950 0.81 ITGB3 (0.42) CNR2CNR1ITGB3ITGAV
SCHEMBL5778333 0.79 CNR1 (0.38) CNR2CNR1ITGB3ITGAVALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0944619-B1 NOVEL INTEGRIN RECEPTOR ANTAGONISTS BRISTOL MYERS SQUIBB PHARMA CO (US) 2006-10-11 EP claimed
EP-0944619-A1 NOVEL INTEGRIN RECEPTOR ANTAGONISTS Du Pont Pharmaceuticals Company (US) 1999-09-29 EP claimed
WO-1998023608-A1 NOVEL INTEGRIN RECEPTOR ANTAGONISTS DUPONT PHARMACEUTICALS COMPANY (US) 1998-06-04 WO claimed
EP-0944619-B1 NOVEL INTEGRIN RECEPTOR ANTAGONISTS BRISTOL MYERS SQUIBB PHARMA CO (US) 2006-10-11 EP disclosed
US-6358976-B1 FOR THERAPY AND PROPHYLAXIS OF CANCER METASTASIS, DIABETIC RETINOPATHY, NEOVASCULAR GLAUCOMA, THROMBOSIS, RESTENOSIS, OSTEOPOROSIS, OR MACULAR DEGENERATION LANTHEUS MI REAL ESTATE, LLC 2002-03-19 US disclosed
US-6130231-A SUBSTITUTED 2,3-DIHYDROQUINOLIN-4-ONES DUPONT PHARMACEUTICALS (US) 2000-10-10 US disclosed
EP-0944619-A1 NOVEL INTEGRIN RECEPTOR ANTAGONISTS Du Pont Pharmaceuticals Company (US) 1999-09-29 EP disclosed
WO-1998023608-A1 NOVEL INTEGRIN RECEPTOR ANTAGONISTS DUPONT PHARMACEUTICALS COMPANY (US) 1998-06-04 WO disclosed