SCHEMBL5779321

SCHEMBL5779321

CC(C)c1csc(C=Cc2cccc(NC(=O)Cc3ccccc3NS(=O)(=O)C(F)(F)F)c2)n1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALB P02768 1/20 0.69
CTPS1 P17812 6/20 0.44
MAPT P10636 3/20 0.41
MEN1 O00255 2/20 0.41
ALDH1A1 P00352 2/20 0.41
TP53 P04637 2/20 0.41
HPGD P15428 2/20 0.41
KMT2A Q03164 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
KDM4E B2RXH2 1/20 0.41
ADRB1 P08588 1/20 0.41
CYP3A4 P08684 1/20 0.41
ADORA3 P0DMS8 1/20 0.41
PTGS1 P23219 1/20 0.41
HSD17B10 Q99714 1/20 0.41
LMNA P02545 2/20 0.35
PTGER3 P43115 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.33
CYSLTR2 Q9NS75 1/20 0.33
CYSLTR1 Q9Y271 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9266527 0.83 ALB (0.83) ALBMAPTMEN1ALDH1A1TP53
SCHEMBL9266539 0.83 ALB (0.83) ALBMAPTMEN1ALDH1A1TP53
SCHEMBL9262889 0.81 ALB (1.00) ALBMAPTMEN1ALDH1A1TP53
SCHEMBL9262876 0.81 ALB (1.00) ALBMAPTMEN1ALDH1A1TP53
SCHEMBL5780400 0.81 ALB (0.53) ALBCTPS1MAPTMEN1ALDH1A1
SCHEMBL9263855 0.79 ALB (0.74) ALBMAPTMEN1ALDH1A1TP53
Acetic Acid SCHEMBL9263847 0.79 ALB (0.75) ALBMAPTMEN1ALDH1A1TP53
Acetic Acid SCHEMBL9263859 0.79 ALB (0.75) ALBMAPTMEN1ALDH1A1TP53
SCHEMBL9264563 0.78 ALB (0.71) ALBCTPS1MAPTMEN1ALDH1A1
SCHEMBL9264552 0.78 ALB (0.71) ALBCTPS1MAPTMEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1652839-A2 Drug efflux pump inhibitor DAIICHI PHARMACEUTICAL CO., LTD. (JP) 2006-05-03 EP disclosed
EP-1227084-B1 DRUG DISCHARGE PUMP INHIBITORS TRINE PHARMACEUTICALS INC (US) 2005-12-14 EP disclosed
EP-1227084-A1 DRUG DISCHARGE PUMP INHIBITORS Microcide Pharmaceuticals, Inc. (US) 2002-07-31 EP disclosed