SCHEMBL5780400

SCHEMBL5780400

CC(C)c1csc(C=Cc2cccc(NC(=O)c3cccc(NS(=O)(=O)C(F)(F)F)c3)c2)n1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALB P02768 1/20 0.53
SNCA P37840 2/20 0.40
ALDH1A1 P00352 3/20 0.39
SMN1; SMN2 Q16637 3/20 0.39
NPC1 O15118 3/20 0.39
RAB9A P51151 3/20 0.39
TP53 P04637 2/20 0.38
KDM4E B2RXH2 1/20 0.38
MEN1 O00255 1/20 0.38
ADRB1 P08588 1/20 0.38
CYP3A4 P08684 1/20 0.38
ADORA3 P0DMS8 1/20 0.38
MAPT P10636 1/20 0.38
HPGD P15428 1/20 0.38
PTGS1 P23219 1/20 0.38
KMT2A Q03164 1/20 0.38
HSD17B10 Q99714 1/20 0.38
PKM P14618 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
CTPS1 P17812 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5779175 0.88 ALB (0.55) ALBSNCAALDH1A1SMN1; SMN2NPC1
SCHEMBL5779321 0.81 ALB (0.69) ALBALDH1A1SMN1; SMN2TP53KDM4E
SCHEMBL5778781 0.80 ALB (0.55) ALBSMN1; SMN2NPC1RAB9AMEN1
SCHEMBL5774563 0.78 ALB (0.69) ALBSNCAALDH1A1SMN1; SMN2NPC1
SCHEMBL27569880 0.78 ALB (0.57) ALBSNCAALDH1A1SMN1; SMN2NPC1
SCHEMBL5780106 0.78 ALB (0.57) ALBSNCAALDH1A1SMN1; SMN2NPC1
SCHEMBL5778029 0.77 ALB (0.51) ALBALDH1A1SMN1; SMN2NPC1RAB9A
SCHEMBL5775071 0.75 ALB (0.60) ALBALDH1A1SMN1; SMN2TP53KDM4E
SCHEMBL5776363 0.74 ALB (0.66) ALBSNCAALDH1A1SMN1; SMN2NPC1
SCHEMBL27588013 0.74 ALB (0.66) ALBSNCAALDH1A1SMN1; SMN2NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1652839-A2 Drug efflux pump inhibitor DAIICHI PHARMACEUTICAL CO., LTD. (JP) 2006-05-03 EP disclosed
EP-1227084-B1 DRUG DISCHARGE PUMP INHIBITORS TRINE PHARMACEUTICALS INC (US) 2005-12-14 EP disclosed
EP-1227084-A1 DRUG DISCHARGE PUMP INHIBITORS Microcide Pharmaceuticals, Inc. (US) 2002-07-31 EP disclosed