SCHEMBL5779344

SCHEMBL5779344

O=Cc1cncc(NC(=O)O)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKT1 P31749 3/20 0.39
ALDH1A1 P00352 3/20 0.37
KDM4E B2RXH2 2/20 0.37
CNR1 P21554 1/20 0.35
NPC1 O15118 2/20 0.33
RAB9A P51151 2/20 0.33
ATM Q13315 1/20 0.33
RAF1 P04049 1/20 0.33
PKM P14618 1/20 0.33
BCAT2 O15382 1/20 0.33
HCAR2 Q8TDS4 1/20 0.32
ROCK2 O75116 1/20 0.32
PIM1 P11309 1/20 0.32
PRKACA P17612 1/20 0.32
FGFR3 P22607 1/20 0.32
GSK3A P49840 1/20 0.32
RPS6KA3 P51812 1/20 0.32
LIMK1 P53667 1/20 0.32
PRKCD Q05655 1/20 0.32
ROCK1 Q13464 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15652470 0.84 LMNA (0.41) AKT1ALDH1A1KDM4ENPC1RAB9A
SCHEMBL23565963 0.76 CLK2 (0.49) ALDH1A1KDM4ENPC1RAB9ADYRK1A
SCHEMBL4069886 0.76 CSF1R (0.47) NAMPT
SCHEMBL2825756 0.76 NAMPT (0.46) RAB9ANAMPT
SCHEMBL3484331 0.75 KDM4E (0.40) ALDH1A1KDM4ECNR1NPC1RAB9A
SCHEMBL1531663 0.75 HCAR2 (0.53) ALDH1A1KDM4EATMHCAR2PRMT5
SCHEMBL15652788 0.75 KDM4E (0.48) ALDH1A1KDM4E
SCHEMBL29957457 0.74 POLB (0.59) ALDH1A1NPC1RAB9AATMROCK2
SCHEMBL4619906 0.73 RXFP1 (0.43) ALDH1A1KDM4ECNR1NPC1RAB9A
SCHEMBL3007374 0.73 POLB (0.52) ALDH1A1KDM4ENPC1RAB9AHCAR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4320132-A1 OXAZEPINE COMPOUNDS AND USES THEREOF IN THE TREATMENT OF CANCER Genentech, Inc. (US) 2024-02-14 EP disclosed
EP-1652839-A2 Drug efflux pump inhibitor DAIICHI PHARMACEUTICAL CO., LTD. (JP) 2006-05-03 EP disclosed
EP-1227084-B1 DRUG DISCHARGE PUMP INHIBITORS TRINE PHARMACEUTICALS INC (US) 2005-12-14 EP disclosed
EP-1227084-A1 DRUG DISCHARGE PUMP INHIBITORS Microcide Pharmaceuticals, Inc. (US) 2002-07-31 EP disclosed