SCHEMBL5779759

SCHEMBL5779759

CC1CN(c2ccc(-c3cc(-c4nncn4-c4cccc(F)c4F)c[nH]3)cn2)CC(C)N1

nearest known ligand 0.36

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 2/20 0.33
HDAC1 Q13547 1/20 0.33
GHSR Q92847 2/20 0.32
TNKS O95271 2/20 0.31
PARP1 P09874 1/20 0.31
PARP15 Q460N3 1/20 0.31
PARP14 Q460N5 1/20 0.31
TNKS2 Q9H2K2 1/20 0.31
PARP2 Q9UGN5 1/20 0.31
SOS1 Q07889 1/20 0.31
SMO Q99835 1/20 0.30
RORC P51449 1/20 0.30
PTPN11 Q06124 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5820058 0.85 CNR2 (0.39) CNR2HDAC1TNKSSOS1
SCHEMBL5781543 0.84 CNR2 (0.52) CNR2
SCHEMBL14002349 0.83 MAP4K1 (0.39)
SCHEMBL4829218 0.83 MAP4K1 (0.39)
SCHEMBL5782679 0.78 TLR7 (0.34)
SCHEMBL5783543 0.75 MELK (0.39) TNKSPARP1TNKS2
SCHEMBL4831565 0.72 MAP4K1 (0.42) CNR2
SCHEMBL5784221 0.70 HCAR1 (0.39)
SCHEMBL5778888 0.70 TNKS (0.42) TNKS
SCHEMBL4824548 0.69 MAP4K1 (0.43) CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1664043-A2 COMPOSITIONS USEFUL AS INHIBITORS OF PROTEIN KINASES Vertex Pharmaceuticals Incorporated (US) 2006-06-07 EP disclosed
WO-2005028475-A2 COMPOSITIONS USEFUL AS INHIBITORS OF PROTEIN KINASES VERTEX PHARMACEUTICALS INCORPORATED (US) 2005-03-31 WO disclosed