SCHEMBL5779807

SCHEMBL5779807

CC(C)c1csc(C=Cc2cccc(C(=O)O)c2)n1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALB P02768 2/20 0.61
TTR P02766 5/20 0.48
UNG P13051 1/20 0.43
FBP1 P09467 1/20 0.43
P4HB P07237 2/20 0.41
HDAC1 Q13547 2/20 0.39
HDAC6 Q9UBN7 2/20 0.39
SLC16A3 O15427 2/20 0.39
NR1H4 Q96RI1 3/20 0.38
HDAC3 O15379 1/20 0.38
HDAC4 P56524 1/20 0.38
HDAC7 Q8WUI4 1/20 0.38
HDAC2 Q92769 1/20 0.38
HDAC10 Q969S8 1/20 0.38
HDAC11 Q96DB2 1/20 0.38
HDAC8 Q9BY41 1/20 0.38
HDAC9 Q9UKV0 1/20 0.38
HDAC5 Q9UQL6 1/20 0.38
NCOR2 Q9Y618 1/20 0.38
PLAU P00749 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27569880 0.87 ALB (0.57) ALBHDAC1HDAC6HDAC3HDAC4
SCHEMBL5780106 0.87 ALB (0.57) ALBHDAC1HDAC6HDAC3HDAC4
SCHEMBL28748039 0.85 ALB (0.54) ALBNR1H4
SCHEMBL5774563 0.82 ALB (0.69) ALBHDAC1HDAC6HDAC3HDAC4
SCHEMBL8304425 0.82 ALB (0.52) ALBUNGHDAC1HDAC6HDAC3
SCHEMBL8304428 0.82 ALB (0.52) ALBUNGHDAC1HDAC6HDAC3
SCHEMBL5775275 0.82 ALB (0.52) ALBFBP1
SCHEMBL7466155 0.80 TTR (0.48) ALBTTRUNGFBP1P4HB
SCHEMBL7466164 0.80 TTR (0.48) ALBTTRUNGFBP1P4HB
SCHEMBL9641854 0.80 ALB (0.49) ALBHDAC1HDAC6NR1H4HDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1652839-A2 Drug efflux pump inhibitor DAIICHI PHARMACEUTICAL CO., LTD. (JP) 2006-05-03 EP disclosed
EP-1227084-B1 DRUG DISCHARGE PUMP INHIBITORS TRINE PHARMACEUTICALS INC (US) 2005-12-14 EP disclosed
EP-1227084-A1 DRUG DISCHARGE PUMP INHIBITORS Microcide Pharmaceuticals, Inc. (US) 2002-07-31 EP disclosed
EP-0287471-B1 CARBOXYSTYRENE DERIVATIVES AND DRUGS CONTAINING THEM AS EFFECTIVE INGREDIENTS MITSUBISHI KASEI CORPORATION (JP) 1992-09-09 EP disclosed
US-4925861-A LEUKOTRIENE ANTAGONISTS, PHOSPHOLIPASE INHIBITORS MITSUBISHI KASEI CORPORATION (JP) 1990-05-15 US disclosed
EP-0287471-A2 Carboxystyrene derivatives and drugs containing them as effective ingredients MITSUBISHI KASEI CORPORATION (JP) 1988-10-19 EP disclosed