SCHEMBL8304425

SCHEMBL8304425

CC(C)c1csc(/C=C/c2cccc(C=O)c2)n1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALB P02768 2/20 0.52
CCR4 P51679 1/20 0.35
HDAC1 Q13547 2/20 0.34
HDAC6 Q9UBN7 2/20 0.34
ALDH1A1 P00352 2/20 0.34
KDM4E B2RXH2 1/20 0.34
MEN1 O00255 1/20 0.34
TP53 P04637 1/20 0.34
ADRB1 P08588 1/20 0.34
CYP3A4 P08684 1/20 0.34
ADORA3 P0DMS8 1/20 0.34
MAPT P10636 1/20 0.34
HPGD P15428 1/20 0.34
PTGS1 P23219 1/20 0.34
KMT2A Q03164 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
HSD17B10 Q99714 1/20 0.34
HDAC3 O15379 1/20 0.33
HDAC4 P56524 1/20 0.33
HDAC7 Q8WUI4 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8304428 1.00 ALB (0.52) ALBCCR4HDAC1HDAC6ALDH1A1
SCHEMBL9641837 0.88 ALB (0.46) ALBMAOAMAOB
SCHEMBL9641842 0.88 ALB (0.46) ALBMAOAMAOB
SCHEMBL9260315 0.83 ALB (0.49) ALBCCR4MAPTMAOAMAOB
SCHEMBL5777449 0.83 ALB (0.49) ALBCCR4MAPTMAOAMAOB
SCHEMBL5775275 0.83 ALB (0.52) ALBMEN1ADORA3PTGS1KMT2A
SCHEMBL5779807 0.82 ALB (0.61) ALBHDAC1HDAC6HDAC3HDAC4
SCHEMBL5776476 0.81 NFE2L2 (0.52) ALBALDH1A1MEN1MAPTKMT2A
SCHEMBL9515918 0.81 NFE2L2 (0.52) ALBALDH1A1MEN1MAPTKMT2A
SCHEMBL8306883 0.80 ALB (0.49) ALBCCR4HDAC1HDAC6ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0469833-B1 N-Benzyl-Indoles, processes for their preparation and pharmaceutical compositions containing them LILLY CO ELI (GB) 1999-09-08 EP disclosed
US-5281593-A Pharmaceuticals LILLY INDUSTRIES LIMITED (GB) 1994-01-25 US disclosed
CN-1061413-A Medicinal compound LILLY INDUSTRIES LTD (GB) 1992-05-27 CN disclosed
EP-0469833-A1 N-Benzyl-Indoles, processes for their preparation and pharmaceutical compositions containing them LILLY INDUSTRIES LIMITED (GB) 1992-02-05 EP disclosed
US-4962117-A ANTIINFLAMMATORY, ANTIASTHMATIC AND CYTOPROTECTIVE AGENTS; ANTIALLERGENS; LEUKOTRIENE ANTAGONISTS MERCK FROSST CANADA, INC. (CA) 1990-10-09 US disclosed
EP-0318085-A2 Heterazole dialkanoic acids MERCK FROSST CANADA INC. (CA) 1989-05-31 EP disclosed