SCHEMBL5780552

SCHEMBL5780552

CN(Cc1ccccc1)C(=O)c1cnc(Nc2cc(Cl)ccc2Cl)nc1C(F)(F)F

nearest known ligand 0.56

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 19/20 0.56
ATF1 P18846 1/20 0.51
NFKB1 P19838 1/20 0.51
CYP1A2 P05177 3/20 0.46
CYP2C9 P11712 3/20 0.46
CYP3A4 P08684 2/20 0.46
CYP2C19 P33261 2/20 0.44
CYP2D6 P10635 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5782167 0.93 CNR2 (0.56) CNR2ATF1NFKB1CYP1A2CYP2C9
SCHEMBL5778821 0.91 CNR2 (0.68) CNR2ATF1NFKB1CYP1A2CYP2C9
SCHEMBL5780255 0.87 CNR2 (0.68) CNR2ATF1NFKB1CYP1A2CYP2C9
SCHEMBL5779533 0.86 CNR2 (0.55) CNR2ATF1NFKB1CYP1A2CYP2C9
SCHEMBL5083384 0.86 CNR2 (0.69) CNR2CYP1A2CYP2C9CYP3A4CYP2C19
SCHEMBL5079708 0.86 CNR2 (0.59) CNR2ATF1NFKB1CYP1A2CYP2C9
SCHEMBL5776710 0.86 CNR2 (0.58) CNR2ATF1NFKB1CYP1A2CYP2C9
SCHEMBL5077147 0.85 CNR2 (0.55) CNR2ATF1NFKB1CYP1A2CYP2C9
SCHEMBL5780683 0.82 CNR2 (0.82) CNR2CYP1A2CYP2C9CYP3A4CYP2C19
SCHEMBL5780970 0.81 CNR2 (0.70) CNR2ATF1NFKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1736470-A2 Pyrimidine derivatives as CB2 cannabinoid receptor modulators GLAXO GROUP LIMITED (GB) 2006-12-27 EP disclosed