SCHEMBL5781663

SCHEMBL5781663

COC(=O)CC(NC(=O)CCCC(=O)O)c1ccc2c(c1)CCCN2

nearest known ligand 0.51

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 20/20 0.51
ITGAV P06756 19/20 0.51
ITGB5 P18084 16/20 0.51
ITGB6 P18564 16/20 0.51
ITGB8 P26012 16/20 0.51
ITGA2B P08514 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5781661 1.00 ITGB3 (0.51) ITGB3ITGAVITGB5ITGB6ITGB8
SCHEMBL5781701 0.94 ITGB3 (0.48) ITGB3ITGAVITGB5ITGB6ITGB8
SCHEMBL5781700 0.94 ITGB3 (0.48) ITGB3ITGAVITGB5ITGB6ITGB8
SCHEMBL5780658 0.79 GAA (0.48) ITGB3ITGAV
SCHEMBL5700994 0.74 TSHR (0.41) ITGB3ITGAVITGB5ITGB6ITGB8
SCHEMBL5700998 0.74 TSHR (0.41) ITGB3ITGAVITGB5ITGB6ITGB8
SCHEMBL5778803 0.71 MAPT (0.54) ITGB3ITGAVITGB5ITGB6ITGB8
SCHEMBL5778799 0.71 MAPT (0.54) ITGB3ITGAVITGB5ITGB6ITGB8
SCHEMBL8333867 0.69 POLB (0.61) ITGB3ITGAVITGB5ITGB6ITGB8
SCHEMBL29679157 0.68 GAA (0.49)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1114028-B1 AZA-BICYCLES WHICH MODULATE THE INHIBITION OF CELL ADHESION AVENTIS PHARMA LTD (GB) 2006-11-29 EP disclosed
US-6608084-B1 Treatment of human or non-human animal patient suffering from, or subject to, condition which can be ameliorated by administration of inhibitor of alpha 4 beta 1 mediated cell adhesion AVENTIS PHARMA LTD. (GB) 2003-08-19 US disclosed
EP-1114028-A1 AZA-BICYCLES WHICH MODULATE THE INHIBITION OF CELL ADHESION Aventis Pharma Limited (GB) 2001-07-11 EP disclosed
WO-2000015612-A1 AZA-BICYCLES WHICH MODULATE THE INHIBITION OF CELL ADHESION AVENTIS PHARMA LIMITED (GB) 2000-03-23 WO disclosed