SCHEMBL578708

SCHEMBL578708

BrNc1cccnc1

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27949708 0.81
SCHEMBL1368828 0.79 KIF11 (0.60)
SCHEMBL29793056 0.79 KIF11 (0.60)
SCHEMBL5266703 0.76
SCHEMBL238813 0.75
SCHEMBL22113986 0.75
SCHEMBL115502 0.75
SCHEMBL4674694 0.75
SCHEMBL14833557 0.75
SCHEMBL1013700 0.75

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 39 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113248426-B Heterocyclic triarylamine compound and organic photoelectric device containing same 浙江华显光电科技有限公司 2024-10-18 CN disclosed
CN-113248426-A Heterocyclic triarylamine compound and organic photoelectric device containing same 浙江华显光电科技有限公司 2021-08-13 CN disclosed
US-10660888-B2 Aminoheteroaryl benzamides as kinase inhibitors NOVARTIS AG (CH) 2020-05-26 US disclosed
US-20190247392-A1 AMINOHETEROARYL BENZAMIDES AS KINASE INHIBITORS NOVARTIS VACCINES AND DIAGNOSTICS, INC. 2019-08-15 US disclosed
US-10188649-B2 Aminoheteroaryl benzamides as kinase inhibitors NOVARTIS AG (CH) 2019-01-29 US disclosed
EP-3063143-B1 AMINOHETEROARYL BENZAMIDES AS KINASE INHIBITORS NOVARTIS AG (CH) 2018-05-16 EP disclosed
US-20180028532-A1 AMINOHETEROARYL BENZAMIDES AS KINASE INHIBITORS NOVARTIS AG (CH) 2018-02-01 US disclosed
US-9763937-B2 Aminoheteroaryl benzamides as kinase inhibitors NOVARTIS AG (CH) 2017-09-19 US disclosed
US-20170182038-A1 AMINOHETEROARYL BENZAMIDES AS KINASE INHIBITORS NOVARTIS AG (CH) 2017-06-29 US disclosed
EP-3063143-A1 AMINOHETEROARYL BENZAMIDES AS KINASE INHIBITORS Novartis AG (CH) 2016-09-07 EP disclosed
US-8481740-B2 Imidazo[1,2 a] pyridine-6-carboxamide derivatives, their use for the treatment of colon cancer and their method of manufacture UNIVERSITY OF THE WITWATERSRAND, JOHANNESBURG (ZA) 2013-07-09 US disclosed
CN-102008459-B Antibacterial agents BIOTA SCIENT MAN 2013-05-29 CN disclosed
CN-101808994-B Compounds and methods for kinase modulation, and indications therefor PLEXXIKON INC 2013-05-15 CN disclosed
CN-103086981-A New compounds NOVARTIS AG 2013-05-08 CN disclosed
US-20120101122-A1 IMIDAZO[1,2 A] PYRIDINE 6 CARBOXAMIDE DERIVATIVES, THEIR USE FOR THE TREATMENT OF COLON CANCER AND THEIR METHOD OF MANUFACTURE UNIVERSITY OF THE WITWATERSRAND, JOHANNESBURG (ZA) 2012-04-26 US disclosed
EP-2417136-A1 IMIDAZ0Ý1,2-A¨PYRIDINE-6-CARBOXAMIDE DERIVATIVES, THEIR USE FOR THE TREATMENT OF COLON CANCER AND THEIR METHOD OF MANUFACTURE University Of Witwatersrand, Johannesburg (ZA) 2012-02-15 EP disclosed
CN-101404989-B Antibacterial agent PROLYSIS LTD 2011-10-05 CN disclosed
CN-102008459-A Antibacterial agents PROLYSIS LTD 2011-04-13 CN disclosed
WO-2010116302-A1 IMIDAZ0[1,2-A] PYRIDINE-6-CARBOXAMIDE DERIVATIVES, THEIR USE FOR THE TREATMENT OF COLON CANCER AND THEIR METHOD OF MANUFACTURE UNIVERSITY OF THE WITWATERSRAND, JOHANNESBURG (ZA) 2010-10-14 WO disclosed
CN-101404989-A Antibacterial agent PROLYSIS LTD (GB) 2009-04-08 CN disclosed