Pyridine

Pyridine

SCHEMBL5787948

c1ccc(COc2cccnc2)cc1.c1ccncc1

nearest known ligand 0.59

Full drug profile on Sugi Atlas →

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 2/20 0.59
MAPT P10636 2/20 0.59
NPSR1 Q6W5P4 1/20 0.59
MAPK1 P28482 2/20 0.58
MEN1 O00255 1/20 0.52
KMT2A Q03164 1/20 0.52
NOS1 P29475 1/20 0.51
NOS2 P35228 1/20 0.51
GRM2 Q14416 2/20 0.50
F2 P00734 1/20 0.49
HTR1A P08908 1/20 0.49
DRD2 P14416 1/20 0.49
P4HTM Q9NXG6 1/20 0.49
CHRNB2 P17787 1/20 0.49
CHRNA4 P43681 1/20 0.49
ALDH1A1 P00352 1/20 0.48
LMNA P02545 1/20 0.48
THRB P10828 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30150593 0.96 RAB9A (0.62) RAB9AMAPTNPSR1MAPK1MEN1
SCHEMBL1323646 0.96 RAB9A (0.62) RAB9AMAPTNPSR1MAPK1MEN1
Bromide SCHEMBL27462942 0.95 RAB9A (0.60) RAB9AMAPTNPSR1MAPK1MEN1
SCHEMBL6238551 0.88 RAB9A (0.55) RAB9AMAPTNPSR1MAPK1MEN1
Acetic Acid SCHEMBL27351298 0.87 KMT2A (0.58) RAB9AMAPTNPSR1MAPK1MEN1
SCHEMBL7539917 0.86 RAB9A (0.60) RAB9AMAPTNPSR1MAPK1MEN1
SCHEMBL7311175 0.85 MAPK1 (0.65) RAB9AMAPK1MEN1KMT2AGRM2
SCHEMBL4313839 0.85 MAPK1 (0.61) RAB9AMAPTNPSR1MAPK1MEN1
Ethoxycarbonyl Group SCHEMBL27686480 0.81 RAB9A (0.51) RAB9AMAPTNPSR1MAPK1MEN1
SCHEMBL24932986 0.81 RAB9A (0.61) RAB9AMAPTNPSR1MAPK1NOS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1664018-A1 BIPYRIDYL AMINES AND ETHERS AS MODULATORS OF METABOTROPIC GLUTAMATE RECEPTOR-5 Merck & Co., Inc. (US) 2006-06-07 EP disclosed
WO-2005021529-A1 BIPYRIDYL AMINES AND ETHERS AS MODULATORS OF METABOTROPIC GLUTAMATE RECEPTOR-5 MERCK & CO., INC. (US) 2005-03-10 WO disclosed