SCHEMBL5788902

SCHEMBL5788902

S=COc1ccc2ccccc2c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 4/20 0.52
CYP1A2 P05177 2/20 0.52
AGXT P21549 2/20 0.47
TDP1 Q9NUW8 3/20 0.45
KDM4E B2RXH2 1/20 0.45
MAPK1 P28482 1/20 0.45
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
CA9 Q16790 1/20 0.44
ALOX5 P09917 1/20 0.44
RELA Q04206 1/20 0.43
PTGS1 P23219 1/20 0.42
GAA P10253 1/20 0.42
RCE1 Q9Y256 1/20 0.42
GPR84 Q9NQS5 1/20 0.42
PTPN7 P35236 1/20 0.41
MEN1 O00255 1/20 0.41
MAPT P10636 1/20 0.41
KMT2A Q03164 1/20 0.41
PPARG P37231 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL97419 0.77 CYP1A2 (0.52) CYP2A6CYP1A2AGXTTDP1KDM4E
SCHEMBL270814 0.77 CYP2A6 (0.58) CYP2A6CYP1A2AGXTTDP1KDM4E
SCHEMBL1225166 0.77 CYP2A6 (0.52) CYP2A6CYP1A2AGXTTDP1KDM4E
SCHEMBL9063781 0.77 CYP2A6 (0.52) CYP2A6CYP1A2AGXTTDP1KDM4E
SCHEMBL3500443 0.75 CYP2A6 (0.67) CYP2A6CYP1A2AGXTTDP1KDM4E
SCHEMBL3306770 0.74 CYP2A6 (0.54) CYP2A6CYP1A2AGXTTDP1KDM4E
SCHEMBL11131812 0.74 CYP1A2 (0.48) CYP2A6CYP1A2AGXTTDP1KDM4E
SCHEMBL9064186 0.74 CYP1A2 (0.48) CYP2A6CYP1A2AGXTTDP1KDM4E
SCHEMBL28546907 0.72 CYP1A2 (0.47) CYP2A6CYP1A2AGXTTDP1KDM4E
SCHEMBL6307841 0.72 CYP2A6 (0.52) CYP2A6CYP1A2AGXTTDP1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115161672-A Method for electrochemically synthesizing amino (dithioperoxy) thiocarbamate compound 广西师范大学 2022-10-11 CN disclosed
EP-1270577-B1 FUROISOQUINOLINE DERIVATIVES, PROCESS FOR PRODUCING THE SAME AND USE THEREOF TAKEDA PHARMACEUTICAL (JP) 2006-12-06 EP disclosed
US-20060106048-A1 Furoisoquinoline derivative and use thereof PASCALI, PETROS P. (CY) 2006-05-18 US disclosed
US-6924292-B2 Furoisoquinoline derivatives, process for producing the same and use thereof TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2005-08-02 US disclosed
EP-1541576-A1 FUROISOQUINOLINE DERIVATIVE AND USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2005-06-15 EP disclosed
US-20040092582-A1 Furoisoquinoline derivatives, process for producing the same and use thereof TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2004-05-13 US disclosed
EP-1270577-A1 FUROISOQUINOLINE DERIVATIVES, PROCESS FOR PRODUCING THE SAME AND USE THEREOF Takeda Chemical Industries, Ltd. (JP) 2003-01-02 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040092582-A1 Furoisoquinoline derivatives, process for producing the same and use thereof PDE3B, PDE5A, PDE3A CYP2A6 1809/4885CYP1A2 399/4885AGXT 3396/4885
US-20060106048-A1 Furoisoquinoline derivative and use thereof PDE3B, PDE2A, PDE3A CYP2A6 326/4885CYP1A2 127/4885AGXT 2420/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.