SCHEMBL5789141

SCHEMBL5789141

COc1cc(C(=O)N2Cc3ccc(C(=O)N(C)CCCN(C)C)n3Cc3ccccc32)ccc1-c1ccccc1

nearest known ligand 0.57

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
AVPR2 P30518 12/20 0.57
AVPR1A P37288 4/20 0.50
ROCK2 O75116 2/20 0.42
PDE4A P27815 1/20 0.39
PDE4B Q07343 1/20 0.39
PDE4C Q08493 1/20 0.39
PDE4D Q08499 1/20 0.39
ROCK1 Q13464 1/20 0.38
PDCD1 Q15116 1/20 0.37
CD274 Q9NZQ7 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5784277 0.93 AVPR2 (0.51) AVPR2AVPR1AROCK2PDE4APDE4B
SCHEMBL5785257 0.93 AVPR2 (0.52) AVPR2AVPR1AROCK2PDE4APDE4B
SCHEMBL5785906 0.91 AVPR2 (0.49) AVPR2AVPR1AROCK2PDE4APDE4B
SCHEMBL5783851 0.91 AVPR1A (0.54) AVPR2AVPR1A
SCHEMBL5785002 0.89 AVPR2 (0.48) AVPR2AVPR1AROCK2PDE4APDE4B
SCHEMBL5784716 0.89 AVPR2 (0.52) AVPR2AVPR1AROCK2PDE4APDE4B
SCHEMBL5787177 0.88 AVPR2 (0.47) AVPR2AVPR1AROCK2PDE4APDE4B
SCHEMBL5786566 0.88 AVPR2 (0.54) AVPR2AVPR1AROCK2PDE4APDE4B
SCHEMBL5784158 0.88 AVPR2 (0.49) AVPR2AVPR1AROCK2PDE4APDE4B
SCHEMBL6632264 0.87 AVPR2 (0.52) AVPR2AVPR1AROCK2PDE4APDE4B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1377586-B1 TRICYCLIC DIAZEPINES AS TOCOLYTIC OXYTOCIN RECEPTOR ANTAGONISTS WYETH CORP (US) 2006-03-22 EP claimed