SCHEMBL5790964

SCHEMBL5790964

COc1ccc(C2=NOC(C)(C(=O)N3CCCC3)C2)cc1C(=O)N1CCC(Cc2ccccc2)CC1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 5/20 0.55
CYP2C9 P11712 4/20 0.55
CYP2C19 P33261 4/20 0.55
MEN1 O00255 6/20 0.45
KMT2A Q03164 6/20 0.45
CYP46A1 Q9Y6A2 1/20 0.45
ALDH1A1 P00352 2/20 0.45
LMNA P02545 2/20 0.45
USP2 O75604 1/20 0.45
TSHR P16473 1/20 0.45
HTT P42858 1/20 0.45
HTR2B P41595 2/20 0.44
PDE4A P27815 1/20 0.44
PDE4B Q07343 1/20 0.44
PDE4C Q08493 1/20 0.44
PDE4D Q08499 1/20 0.44
APOBEC3A P31941 1/20 0.42
APOBEC3G Q9HC16 1/20 0.42
ACHE P22303 1/20 0.42
MGLL Q99685 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5792778 0.90 MAPK14 (0.57) MAPK14CYP2C9CYP2C19MEN1KMT2A
SCHEMBL5789441 0.89 MAPK14 (0.50) MAPK14CYP2C9CYP2C19MEN1KMT2A
SCHEMBL3549439 0.85 PDE4B (0.62) MAPK14CYP2C9CYP2C19MEN1KMT2A
SCHEMBL5791454 0.85 HTT (0.52) MAPK14CYP2C9CYP2C19MEN1KMT2A
SCHEMBL5789709 0.84 HTT (0.51) MAPK14CYP2C9CYP2C19MEN1KMT2A
SCHEMBL5792828 0.83 CYP2C9 (0.53) MAPK14CYP2C9CYP2C19MEN1KMT2A
SCHEMBL5792547 0.82 MAPK14 (0.55) MAPK14CYP2C9CYP2C19ALDH1A1LMNA
SCHEMBL5807168 0.82 MAPK14 (0.55) MAPK14CYP2C9CYP2C19ALDH1A1LMNA
SCHEMBL5791336 0.81 MAPK14 (0.49) MAPK14CYP2C9CYP2C19ALDH1A1LMNA
SCHEMBL5790812 0.78 GAA (0.57) MAPK14CYP2C9CYP2C19MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006016237-A2 HETEROCYCLIC DERIVATIVES AS ANTI-INFLAMMATORY AGENTS RANBAXY LABORATORIES LIMITED (IN) 2006-02-16 WO disclosed