SCHEMBL5793017

SCHEMBL5793017

CNc1nc2ccc([N+](=O)[O-])cc2s1.Nc1ccccc1NC(=O)c1ccccc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 5/20 0.58
RAB9A P51151 4/20 0.58
MCL1 Q07820 1/20 0.58
SMN1; SMN2 Q16637 4/20 0.56
LMNA P02545 3/20 0.56
S1PR2 O95136 1/20 0.56
NPY1R P25929 1/20 0.56
HTT P42858 1/20 0.56
NPY2R P49146 1/20 0.56
NPSR1 Q6W5P4 1/20 0.56
DYRK1A Q13627 1/20 0.55
MAPT P10636 4/20 0.54
ALDH1A1 P00352 3/20 0.54
MMP13 P45452 2/20 0.53
SCD O00767 2/20 0.53
KMT2A Q03164 5/20 0.53
MEN1 O00255 4/20 0.53
HDAC1 Q13547 2/20 0.52
POLB P06746 2/20 0.52
STAT1 P42224 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL211614 0.84 HDAC1 (0.74) NPC1RAB9AMCL1SMN1; SMN2LMNA
SCHEMBL2187627 0.84 NPC1 (0.80) NPC1RAB9AMCL1SMN1; SMN2LMNA
SCHEMBL4914634 0.80 NPC1 (0.74) NPC1RAB9AMCL1SMN1; SMN2LMNA
SCHEMBL3753095 0.79 DYRK1A (0.71) NPC1RAB9AMCL1SMN1; SMN2LMNA
SCHEMBL16562175 0.76 NPC1 (0.79) NPC1RAB9AMCL1SMN1; SMN2LMNA
SCHEMBL7128296 0.75 NPC1 (0.77) NPC1RAB9AMCL1SMN1; SMN2LMNA
SCHEMBL19174351 0.75 HDAC2 (0.76) NPC1RAB9ASMN1; SMN2HTTMAPT
SCHEMBL2189310 0.75 SCD (0.74) NPC1RAB9AMCL1SMN1; SMN2LMNA
SCHEMBL2191669 0.74 NPC1 (1.00) NPC1RAB9AMCL1SMN1; SMN2LMNA
SCHEMBL16684914 0.74 HDAC1 (0.73) NPC1RAB9AMAPTALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1735319-A1 INHIBITORS OF HISTONE DEACETYLASE Methylgene, Inc. (CA) 2006-12-27 EP disclosed
WO-2005092899-A1 INHIBITORS OF HISTONE DEACETYLASE METHYLGENE INC. (CA) 2005-10-06 WO disclosed