SCHEMBL5793280

SCHEMBL5793280

O=C(c1cccc(CCCN2CCOCC2)c1)c1c[nH]nc1-c1ccc(F)cc1F

nearest known ligand 0.57

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 5/20 0.57
KMT2A Q03164 1/20 0.41
EPHX2 P34913 4/20 0.41
PARP1 P09874 2/20 0.41
FFAR1 O14842 1/20 0.40
DRD2 P14416 1/20 0.39
SLC6A4 P31645 1/20 0.39
SLC6A3 Q01959 1/20 0.39
POLB P06746 1/20 0.39
SIGMAR1 Q99720 1/20 0.39
BCL3 P20749 1/20 0.39
PCSK9 Q8NBP7 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7809769 0.88 MAPK14 (0.61) MAPK14EPHX2PARP1POLBSIGMAR1
SCHEMBL5323843 0.84 MAPK14 (0.56) MAPK14KMT2AEPHX2PARP1FFAR1
SCHEMBL1384090 0.76 MAPK14 (0.80) MAPK14
SCHEMBL5322574 0.74 MAPK14 (0.61) MAPK14EPHX2PARP1POLBSIGMAR1
Hydrochloric Acid SCHEMBL7468024 0.73 MAPK14 (0.60) MAPK14EPHX2PARP1POLBSIGMAR1
SCHEMBL7475922 0.73 MAPK14 (0.44) MAPK14KMT2ADRD2SLC6A4SLC6A3
SCHEMBL1385480 0.72 MAPK14 (1.00) MAPK14
Hydrochloric Acid SCHEMBL7812345 0.72 MAPK14 (0.62) MAPK14EPHX2
Hydrochloric Acid SCHEMBL6157505 0.72 MAPK14 (0.98) MAPK14
Hydrochloric Acid SCHEMBL7809765 0.70 MAPK14 (0.67) MAPK14EPHX2POLBSIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1641764-A1 5-MEMBERED HETEROCYCLE-BASED P38 KINASE INHIBITORS Novartis AG (CH) 2006-04-05 EP disclosed
WO-2005009973-A1 5-MEMBERED HETEROCYCLE-BASED P38 KINASE INHIBITORS NOVARTIS AG (CH) 2005-02-03 WO disclosed