SCHEMBL7475922

SCHEMBL7475922

Nc1[nH]nc(-c2ccc(F)cc2F)c1C(=O)c1cccc(CCCN2CCS(=O)(=O)CC2)c1

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 5/20 0.44
SLC6A4 P31645 2/20 0.38
DRD2 P14416 1/20 0.38
SLC6A3 Q01959 1/20 0.38
KIF11 P52732 1/20 0.35
ALOX15 P16050 1/20 0.35
GAA P10253 2/20 0.35
SIGMAR1 Q99720 2/20 0.34
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
MAPK8 P45983 1/20 0.33
MAPK10 P53779 1/20 0.33
ALDH1A1 P00352 2/20 0.33
HTT P42858 1/20 0.33
LMNA P02545 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5323843 0.89 MAPK14 (0.56) MAPK14SLC6A4DRD2SLC6A3KIF11
SCHEMBL7803286 0.81 MAPK14 (0.54) MAPK14SLC6A4DRD2SLC6A3SIGMAR1
SCHEMBL7475964 0.80 CYP2D6 (0.47) ALOX15GAAALDH1A1HTTLMNA
SCHEMBL7482460 0.79 MAPK14 (0.53) MAPK14ALOX15MAPK8MAPK10
SCHEMBL5322574 0.78 MAPK14 (0.61) MAPK14GAASIGMAR1ALDH1A1LMNA
SCHEMBL7481210 0.77 PTAFR (0.42) MAPK14ALOX15ALDH1A1HTT
Hydrochloric Acid SCHEMBL7468024 0.77 MAPK14 (0.60) MAPK14SIGMAR1
SCHEMBL6160299 0.75 MAPK14 (0.64) MAPK14
SCHEMBL7464576 0.73 ALOX15 (0.47) MAPK14ALOX15KMT2AMAPK10
SCHEMBL7474793 0.73 ALOX15 (0.44) MAPK14ALOX15GAAMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1218346-A1 PYRAZOLE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2002-07-03 EP disclosed
WO-2001021591-A1 PYRAZOLE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2001-03-29 WO disclosed