SCHEMBL5794589

SCHEMBL5794589

COc1cc2c(-c3ccc[nH]3)cn(CCCN3CCCN(C)CC3)c2cc1OC

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 3/20 0.46
GSK3B P49841 3/20 0.46
HTR1A P08908 1/20 0.38
DRD2 P14416 1/20 0.38
SLC6A2 P23975 1/20 0.38
HTR2A P28223 1/20 0.38
SLC6A4 P31645 1/20 0.38
DRD3 P35462 1/20 0.38
SLC6A3 Q01959 1/20 0.38
FLT1 P17948 1/20 0.37
FLT4 P35916 1/20 0.37
PRKCB P05771 1/20 0.37
PRKCA P17252 1/20 0.37
HTR7 P34969 1/20 0.37
QPCT Q16769 2/20 0.37
FLT3 P36888 1/20 0.36
MEN1 O00255 1/20 0.35
POLB P06746 1/20 0.35
KMT2A Q03164 1/20 0.35
EHMT2 Q96KQ7 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5795129 0.90 GSK3B (0.42) KDRGSK3BHTR1ADRD2SLC6A2
SCHEMBL1748879 0.81 IGF1R (0.61) KDRGSK3BDRD2DRD3QPCT
SCHEMBL5794829 0.80 IGF1R (0.39) KDRGSK3BHTR1ADRD2SLC6A2
SCHEMBL5798073 0.78 IGF1R (0.45) KDRFLT1FLT4
SCHEMBL5794484 0.78 IGF1R (0.40) GSK3BMEN1KMT2A
SCHEMBL1748413 0.75 IGF1R (0.63) KDRGSK3BDRD2DRD3HTR7
Trifluoroacetic Acid SCHEMBL1748997 0.75 IGF1R (0.53) KDRGSK3BDRD2DRD3PRKCB
SCHEMBL5821747 0.74 HTR6 (0.44) KDRGSK3BKMT2A
SCHEMBL5794491 0.73 GSK3B (0.39) KDRGSK3BHTR1ADRD2SLC6A2
SCHEMBL5795213 0.73 KDR (0.37) KDRGSK3BFLT1FLT4HTR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1732546-A2 NOVEL PYRROLO (2,3-B)PYRIDINE DERIVATIVES, THE PREPARATION AND THE PHARMACEUTICAL USE THEREOF IN THE FORM OF KINASE INHIBITORS Aventis Pharma S.A. (FR) 2006-12-20 EP disclosed
WO-2005095399-A2 NOVEL PYRROLO (2,3-B)PYRIDINE DERIVATIVES, THE PREPARATION AND THE PHARMACEUTICAL USE THEREOF IN THE FORM OF KINASE INHIBITORS AVENTIS PHARMA S.A. (FR) 2005-10-13 WO disclosed