SCHEMBL5794986

SCHEMBL5794986

C=COC(=O)OCc1ccsc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC1A3 P43003 2/20 0.43
SLC1A2 P43004 2/20 0.43
SLC1A1 P43005 2/20 0.43
CYP1A2 P05177 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.36
ENPP2 Q13822 1/20 0.35
ATXN2 Q99700 1/20 0.35
PARP15 Q460N3 1/20 0.35
PARP10 Q53GL7 1/20 0.35
PARP3 Q9Y6F1 1/20 0.35
HPGD P15428 2/20 0.35
TAAR1 Q96RJ0 1/20 0.34
HDAC8 Q9BY41 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
ALDH1A1 P00352 1/20 0.34
THRB P10828 1/20 0.34
HTT P42858 1/20 0.34
MAPT P10636 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9903115 0.80 SLC1A3 (0.45) SLC1A3SLC1A2SLC1A1CYP1A2CYP2C9
SCHEMBL13788676 0.77 SLC1A3 (0.43) SLC1A3SLC1A2SLC1A1CYP1A2CYP2C9
SCHEMBL8129509 0.76 MEN1 (0.52)
SCHEMBL5793033 0.76 ALDH1A1 (0.53) L3MBTL1ALDH1A1
SCHEMBL5794984 0.74 SLC1A3 (0.40) SLC1A3SLC1A2SLC1A1CYP1A2CYP2C9
SCHEMBL13044441 0.74 ALDH1A1 (0.55) SLC1A3SLC1A2SLC1A1CYP1A2CYP2C9
SCHEMBL7652109 0.74 SLC1A3 (0.53) SLC1A3SLC1A2SLC1A1CYP1A2CYP2C9
SCHEMBL13170592 0.74 SLC1A3 (0.49) SLC1A3SLC1A2SLC1A1CYP1A2CYP2C9
Hydrochloric Acid SCHEMBL27717048 0.73 ALDH1A1 (0.53) SLC1A3SLC1A2SLC1A1CYP1A2CYP2C9
SCHEMBL9075028 0.72 SLC1A3 (0.44) SLC1A3SLC1A2SLC1A1CYP1A2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003057896-A1 METHODS FOR PREPARING ANTHRACYCLINONE DERIVATIVES AND ANTHRACYCLINONE DERIVATIVES PER SE ALBANY MOLECULAR RESEARCH, INC. (US) 2003-07-17 WO claimed
WO-2003057687-A1 METHODS FOR PREPARING DOXORUBICIN DERIVATIVES ALBANY MOLECULAR RESEARCH, INC. (US) 2003-07-17 WO claimed
WO-2006012277-A2 BIOCATALYTIC PROCESS FOR PREPARING ENANTIOMERICALLY ENRICHED PRAMIPEXOLE AMR TECHNOLOGY, INC. (US) 2006-02-02 WO disclosed
WO-2003057896-A1 METHODS FOR PREPARING ANTHRACYCLINONE DERIVATIVES AND ANTHRACYCLINONE DERIVATIVES PER SE ALBANY MOLECULAR RESEARCH, INC. (US) 2003-07-17 WO disclosed
WO-2003057687-A1 METHODS FOR PREPARING DOXORUBICIN DERIVATIVES ALBANY MOLECULAR RESEARCH, INC. (US) 2003-07-17 WO disclosed