SCHEMBL5795340

SCHEMBL5795340

CNc1nn2c(=O)n(Cc3ccc(CC(F)(F)F)cc3)nc2c(-c2ccc(Cl)cc2)c1-c1ccc(Cl)cc1

nearest known ligand 0.52

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 18/20 0.52
CYP3A4 P08684 4/20 0.39
CYP2C9 P11712 3/20 0.39
CYP2C19 P33261 3/20 0.39
HTT P42858 1/20 0.34
LMNA P02545 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3561075 0.90 CNR1 (0.57) CNR1CYP3A4CYP2C9CYP2C19LMNA
SCHEMBL13134239 0.89 CNR1 (0.50) CNR1CYP3A4CYP2C9CYP2C19HTT
SCHEMBL13114733 0.87 CNR1 (0.51) CNR1CYP3A4CYP2C19NPSR1
SCHEMBL5796174 0.86 CNR1 (0.54) CNR1CYP3A4CYP2C9CYP2C19HTT
SCHEMBL5795343 0.84 CNR1 (0.47) CNR1CYP3A4CYP2C9CYP2C19LMNA
SCHEMBL13114664 0.80 CNR1 (0.54) CNR1CYP3A4CYP2C9CYP2C19LMNA
SCHEMBL13114655 0.76 CNR1 (0.51) CNR1CYP3A4CYP2C9CYP2C19LMNA
SCHEMBL4806813 0.76 CNR1 (0.73) CNR1CYP3A4CYP2C9CYP2C19HTT
SCHEMBL3550428 0.75 CNR1 (0.59) CNR1CYP3A4CYP2C9CYP2C19LMNA
SCHEMBL13114662 0.74 CNR1 (0.58) CNR1CYP3A4CYP2C9CYP2C19LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1697371-A1 AZABICYCLIC HETEROCYCLES AS CANNABINOID RECEPTOR MODULATORS Bristol-Myers Squibb Company (US) 2006-09-06 EP disclosed
WO-2005063762-A1 AZABICYCLIC HETEROCYCLES AS CANNABINOID RECEPTOR MODULATORS BRISTOL-MYERS SQUIBB COMPANY (US) 2005-07-14 WO disclosed