SCHEMBL5796552

SCHEMBL5796552

COc1cc2c(-c3ccc(F)[nH]3)cn(CCN3CCOCC3)c2cc1OC

nearest known ligand 0.45

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KDR P35968 1/20 0.45
GSK3B P49841 1/20 0.45
KDM4E B2RXH2 2/20 0.43
RCE1 Q9Y256 1/20 0.43
MAPK1 P28482 2/20 0.42
CNR1 P21554 2/20 0.41
DRD2 P14416 1/20 0.41
DRD3 P35462 1/20 0.41
CCNT1 O60563 4/20 0.41
CDK9 P50750 4/20 0.41
CNR2 P34972 3/20 0.41
MKNK2 Q9HBH9 1/20 0.39
SYK P43405 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5794491 0.91 GSK3B (0.39) KDRGSK3BKDM4ERCE1DRD2
SCHEMBL5797776 0.84 KDM4E (0.44) KDRGSK3BKDM4ERCE1MAPK1
SCHEMBL5793991 0.79 KDR (0.43) KDRGSK3BKDM4ERCE1MAPK1
SCHEMBL1748831 0.79 IGF1R (0.46) KDRGSK3BKDM4ERCE1MAPK1
SCHEMBL1779928 0.78 IGF1R (0.66) KDRGSK3BKDM4ERCE1CNR1
SCHEMBL1749184 0.78 CDK9 (0.43) KDRKDM4ERCE1CCNT1CDK9
SCHEMBL1748609 0.77 CDK9 (0.47) KDRGSK3BKDM4ERCE1CCNT1
SCHEMBL5797872 0.77 IGF1R (0.55) KDRGSK3BKDM4ECDK9
SCHEMBL5795129 0.72 GSK3B (0.42) KDRGSK3BCNR1DRD2DRD3
SCHEMBL5822423 0.72 TP53 (0.43) KDRGSK3BKDM4ERCE1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1732546-A2 NOVEL PYRROLO (2,3-B)PYRIDINE DERIVATIVES, THE PREPARATION AND THE PHARMACEUTICAL USE THEREOF IN THE FORM OF KINASE INHIBITORS Aventis Pharma S.A. (FR) 2006-12-20 EP disclosed
WO-2005095399-A2 NOVEL PYRROLO (2,3-B)PYRIDINE DERIVATIVES, THE PREPARATION AND THE PHARMACEUTICAL USE THEREOF IN THE FORM OF KINASE INHIBITORS AVENTIS PHARMA S.A. (FR) 2005-10-13 WO disclosed