SCHEMBL5797110

SCHEMBL5797110

Cc1c(CC(=O)O)c2c(F)c(OC(=O)C(c3c(C)n(C(=O)c4ccc(Cl)cc4)c4cc(F)c(O)c(F)c34)C(C)(C)C)c(F)cc2n1C(=O)c1ccc(Cl)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 4/20 0.47
AKR1C2 P52895 4/20 0.47
PTGS2 P35354 7/20 0.45
PTGS1 P23219 5/20 0.45
ABCB1 P08183 4/20 0.43
GLO1 Q04760 2/20 0.43
HIF1A Q16665 2/20 0.43
KDM4E B2RXH2 1/20 0.43
MEN1 O00255 1/20 0.43
PTGES O14684 1/20 0.43
ABCC3 O15438 1/20 0.43
ABCC4 O15439 1/20 0.43
ABCB11 O95342 1/20 0.43
MT-CO2 P00403 1/20 0.43
LMNA P02545 1/20 0.43
ALB P02768 1/20 0.43
CYP1A2 P05177 1/20 0.43
ALOX5 P09917 1/20 0.43
ADORA3 P0DMS8 1/20 0.43
CXCL8 P10145 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5796936 0.92 AKR1C3 (0.39) AKR1C3AKR1C2PTGS2PTGS1ABCB1
SCHEMBL5798705 0.86 AKR1C3 (0.45) AKR1C3AKR1C2PTGS2PTGS1ABCB1
SCHEMBL5554506 0.83 AKR1C3 (0.64) AKR1C3AKR1C2PTGS2PTGS1ABCB1
SCHEMBL5796494 0.83 AKR1C3 (0.40) AKR1C3AKR1C2PTGS2PTGS1ABCB1
SCHEMBL5800198 0.82 AKR1C3 (0.39) AKR1C3AKR1C2PTGS2PTGS1ABCB1
SCHEMBL6424132 0.82 AKR1C3 (0.41) AKR1C3AKR1C2PTGS2PTGS1ABCB1
SCHEMBL5797960 0.79 AKR1C3 (0.38) AKR1C3AKR1C2PTGS2PTGS1ABCB1
SCHEMBL5798581 0.79 AKR1C3 (0.38) AKR1C3AKR1C2PTGS2PTGS1ABCB1
SCHEMBL5800670 0.79 PTGS2 (0.60) AKR1C3AKR1C2PTGS2PTGS1ABCB1
SCHEMBL5801056 0.79 AKR1C3 (0.37) AKR1C3AKR1C2PTGS2PTGS1ABCB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006050120-A2 SYNTHESIS OF COX-2 AND FAAH INHIBITORS MICROBIA, INC. (US) 2006-05-11 WO disclosed