SCHEMBL5798677

SCHEMBL5798677

CC(=O)OC/C(=C(\CO)c1ccc(F)c(F)c1)c1ccc(S(C)(=O)=O)cc1

nearest known ligand 0.47

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 9/20 0.45
ESR2 Q92731 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3867297 0.88 ESR2 (0.52) PTGS2ESR2
SCHEMBL3867288 0.88 ESR2 (0.52) PTGS2ESR2
SCHEMBL3868554 0.88 ESR2 (0.52) PTGS2ESR2
SCHEMBL3868550 0.88 ESR2 (0.52) PTGS2ESR2
SCHEMBL5807999 0.87 PTGS2 (0.52) PTGS2ESR2
SCHEMBL3480155 0.87 PTGS2 (0.52) PTGS2ESR2
SCHEMBL3480153 0.87 PTGS2 (0.52) PTGS2ESR2
SCHEMBL5798485 0.85 PTGS2 (0.45) PTGS2ESR2
SCHEMBL3480364 0.85 PTGS2 (0.45) PTGS2ESR2
SCHEMBL3480365 0.85 PTGS2 (0.45) PTGS2ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0788476-B1 STILBENE DERIVATIVES USEFUL AS CYCLOOXYGENASE-2 INHIBITORS MERCK FROSST CANADA INC (CA) 1999-10-20 EP claimed
WO-2006044230-A1 WATER SOLUBLE PRODRUGS OF COX-2 INHIBITORS MERCK & CO., INC. (US) 2006-04-27 WO disclosed
US-5849943-A Stilbene derivatives useful as cyclooxygenase-2 inhibitors MERCK FROSST CANADA, INC. (CA) 1998-12-15 US disclosed