SCHEMBL5799073

SCHEMBL5799073

CC(C)CC(O)(Cc1cc2cnccc2s1)C(F)F

nearest known ligand 0.48

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 5/20 0.48
NR3C1 P04150 1/20 0.36
PGR P06401 1/20 0.36
NR3C2 P08235 1/20 0.36
MET P08581 1/20 0.32
KDM4C Q9H3R0 1/20 0.32
TGFBR1 P36897 1/20 0.32
LNPEP Q9UIQ6 1/20 0.30
OGA O60502 1/20 0.30
HDAC3 O15379 1/20 0.30
HDAC1 Q13547 1/20 0.30
HDAC2 Q92769 1/20 0.30
NCOR2 Q9Y618 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3714152 0.73 NR3C1 (0.47) NR3C1PGRNR3C2
SCHEMBL2176886 0.69 CYP2A6 (0.69) CYP2A6METKDM4CTGFBR1HDAC3
SCHEMBL10653557 0.69 CYP2A6 (0.69) CYP2A6METKDM4CTGFBR1HDAC3
SCHEMBL12487353 0.66 CYP2A6 (1.00) CYP2A6METKDM4CTGFBR1
SCHEMBL1251644 0.66 CYP2A6 (1.00) CYP2A6METKDM4CTGFBR1HDAC3
SCHEMBL27168295 0.66 CYP2A6 (0.63) CYP2A6METKDM4CTGFBR1HDAC3
SCHEMBL30048549 0.66 CYP2A6 (0.63) CYP2A6KDM4CHDAC3HDAC1HDAC2
Hydrochloric Acid SCHEMBL2179295 0.65 CYP2A6 (0.96) CYP2A6MET
Hydrochloric Acid SCHEMBL31751429 0.65 CYP2A6 (0.96) CYP2A6MET
SCHEMBL291661 0.64 NR3C1 (0.66) NR3C1PGRNR3C2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1673088-A1 1,1,1- TRIFLUORO-4-PHENYL-4-METHYL-2-(1H-PYRROLO¬2,3-C|PYRIDIN-2-YLMETHYL)PENTAN-2-OL DERIVATIVES AND RELATED COMPOUNDS AS GLUCOCORTICOID LIGANDS FOR THE TREATMENT OF INFLAMMATORY DISEASES AND DIABETES BOEHRINGER INGELHEIM PHARMACEUTICALS INC. (US) 2006-06-28 EP disclosed
WO-2005030213-A1 1,1,1-TRIFLUORO-4-PHENYL-4-METHYL-2-(1H-PYRROLO BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2005-04-07 WO disclosed