SCHEMBL5800145

SCHEMBL5800145

CCC(C)NC(=O)Cc1c(C)n(C(=O)c2cccc(Cl)c2)c2cc(F)c(O)c(F)c12.CCCCNC(=O)Cc1c(C)n(C(=O)c2cccc(Cl)c2)c2cc(F)c(O)c(F)c12

nearest known ligand 0.46

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 17/20 0.46
PTGS1 P23219 4/20 0.41
HRH4 Q9H3N8 1/20 0.40
HDAC3 O15379 3/20 0.39
HDAC1 Q13547 3/20 0.39
HDAC8 Q9BY41 3/20 0.39
HDAC6 Q9UBN7 3/20 0.39
HDAC2 Q92769 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5559027 0.93 PTGS2 (0.51) PTGS2
SCHEMBL5553613 0.93 PTGS2 (0.49) PTGS2PTGS1HRH4HDAC3HDAC1
SCHEMBL5559021 0.93 PTGS2 (0.51) PTGS2
SCHEMBL5798070 0.91 PTGS2 (0.47) PTGS2PTGS1HRH4HDAC3HDAC1
SCHEMBL5558568 0.88 PTGS2 (0.45) PTGS2PTGS1HRH4HDAC3HDAC1
SCHEMBL5800149 0.87 PTGS2 (0.42) PTGS2PTGS1HRH4HDAC3HDAC1
SCHEMBL5554016 0.85 PTGS2 (0.48) PTGS2
SCHEMBL5554009 0.85 PTGS2 (0.48) PTGS2
SCHEMBL5554400 0.85 PTGS2 (0.44) PTGS2PTGS1HRH4HDAC3HDAC1
SCHEMBL5559464 0.85 TP53 (0.42) PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006050120-A2 SYNTHESIS OF COX-2 AND FAAH INHIBITORS MICROBIA, INC. (US) 2006-05-11 WO disclosed