SCHEMBL5800267

SCHEMBL5800267

CC(C)(C)OC(=O)Nc1ccc(F)cc1O

nearest known ligand 0.51

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KCNQ4 P56696 3/20 0.51
KCNQ5 Q9NR82 3/20 0.51
CYP17A1 P05093 1/20 0.44
RXFP1 Q9HBX9 1/20 0.41
POLB P06746 2/20 0.40
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
HDAC3 O15379 1/20 0.40
HDAC1 Q13547 1/20 0.40
MAPT P10636 1/20 0.40
HTT P42858 1/20 0.40
KCNMA1 Q12791 1/20 0.39
PLA2G7 Q13093 1/20 0.39
LMNA P02545 1/20 0.39
HSP90AA1 P07900 1/20 0.38
HSP90AB1 P08238 1/20 0.38
BRD9 Q9H8M2 1/20 0.38
GAA P10253 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL857284 0.86 HTT (0.55) KCNQ4KCNQ5CYP17A1POLBNPC1
SCHEMBL8292291 0.84 KCNQ4 (0.48) KCNQ4KCNQ5CYP17A1MAPTHTT
SCHEMBL2391319 0.84 CXCR2 (0.53) POLBNPC1RAB9AMAPTLMNA
SCHEMBL197145 0.83 HDAC1 (0.55) KCNQ4KCNQ5CYP17A1HDAC3HDAC1
SCHEMBL16692867 0.83 KCNQ4 (0.47) KCNQ4KCNQ5CYP17A1RXFP1POLB
SCHEMBL22092641 0.83 KCNQ4 (0.47) KCNQ4KCNQ5CYP17A1RXFP1POLB
SCHEMBL29581478 0.83 HDAC1 (0.55) KCNQ4KCNQ5CYP17A1HDAC3HDAC1
SCHEMBL26426327 0.83 KCNQ4 (0.50) KCNQ4KCNQ5CYP17A1RXFP1POLB
SCHEMBL13055401 0.83 CA12 (0.49) KCNQ4KCNQ5CYP17A1RXFP1POLB
SCHEMBL15614546 0.83 MAPT (0.51) KCNQ4KCNQ5CYP17A1RXFP1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106458969-A (substituted phenyl) (substituted pyrimidine) amino derivative and preparation method and pharmaceutical application thereof 四川海思科制药有限公司 2017-02-22 CN disclosed
WO-2016029839-A1 (SUBSTITUTED PHENYL) (SUBSTITUTED PYRIMIDINE) AMINO DERIVATIVE, PREPARATION METHOD THEREFOR, AND MEDICATION USE 四川海思科制药有限公司 2016-03-03 WO disclosed
WO-2006071035-A1 NOVEL ([1,3]THIAZOLO[5,4-B]PYRIDIN-2-YL)-2-CARBOXAMIDE DERIVATIVES LG LIFE SCIENCES, LTD. (KR) 2006-07-06 WO disclosed