SCHEMBL5800980

SCHEMBL5800980

COc1ccc(F)cc1C(C)(C)CC(O)(Cc1ccnc(C#N)c1)C(F)F

nearest known ligand 0.52

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
NR3C1 P04150 20/20 0.52
NR3C2 P08235 12/20 0.52
PGR P06401 6/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL291256 0.87 NR3C1 (0.70) NR3C1NR3C2PGR
SCHEMBL27754173 0.80 NR3C1 (0.58) NR3C1NR3C2PGR
SCHEMBL27754175 0.77 NR3C1 (0.52) NR3C1NR3C2PGR
SCHEMBL1634849 0.73 NR3C1 (0.71) NR3C1NR3C2PGR
SCHEMBL5821253 0.72 NR3C1 (0.41) NR3C1NR3C2PGR
SCHEMBL1634553 0.71 NR3C1 (0.68) NR3C1NR3C2PGR
SCHEMBL1635059 0.71 NR3C1 (0.72) NR3C1NR3C2PGR
SCHEMBL293361 0.70 NR3C1 (0.78) NR3C1NR3C2PGR
SCHEMBL300174 0.70 NR3C1 (0.86) NR3C1NR3C2PGR
SCHEMBL292014 0.69 NR3C1 (0.75) NR3C1NR3C2PGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1673088-A1 1,1,1- TRIFLUORO-4-PHENYL-4-METHYL-2-(1H-PYRROLO¬2,3-C|PYRIDIN-2-YLMETHYL)PENTAN-2-OL DERIVATIVES AND RELATED COMPOUNDS AS GLUCOCORTICOID LIGANDS FOR THE TREATMENT OF INFLAMMATORY DISEASES AND DIABETES BOEHRINGER INGELHEIM PHARMACEUTICALS INC. (US) 2006-06-28 EP disclosed
WO-2005030213-A1 1,1,1-TRIFLUORO-4-PHENYL-4-METHYL-2-(1H-PYRROLO BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2005-04-07 WO disclosed