SCHEMBL5801334

SCHEMBL5801334

CNC(C)C(=O)OC.COC(=O)C(C)NCCC(=O)OC(C)(C)C

nearest known ligand 0.40

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CA14 Q9ULX7 3/20 0.40
CA12 O43570 2/20 0.40
CA1 P00915 2/20 0.34
CA2 P00918 2/20 0.34
CYP2D6 P10635 1/20 0.33
EPHX2 P34913 1/20 0.31
MLYCD O95822 1/20 0.30
CA7 P43166 1/20 0.30
TSHR P16473 1/20 0.30
DGAT1 O75907 1/20 0.30
HDAC3 O15379 1/20 0.30
HDAC1 Q13547 1/20 0.30
HDAC2 Q92769 1/20 0.30
HDAC8 Q9BY41 1/20 0.30
HDAC6 Q9UBN7 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3202642 0.94 CA14 (0.44) CA14CA12CA1CA2CYP2D6
SCHEMBL2324579 0.82 MEN1 (0.40) CA14CA12CA1CA2CYP2D6
SCHEMBL3193199 0.82 MEN1 (0.40) CA14CA12CA1CA2CYP2D6
SCHEMBL3670762 0.78 CYP2D6 (0.41) CA14CA12CA1CA2CYP2D6
SCHEMBL7431200 0.77 CA14 (0.46) CA14CA12CA1CA2CYP2D6
SCHEMBL4095492 0.77 CA14 (0.46) CA14CA12CA1CA2CYP2D6
SCHEMBL29023037 0.74 GAA (0.45) CA14TSHR
SCHEMBL5801336 0.74 CA14 (0.46) CA14CA12CA1CA2CA7
SCHEMBL13613755 0.74 CA12 (0.44) CA14CA12CA1CA2CA7
SCHEMBL14206399 0.73 CA12 (0.50) CA14CA12CA1CA2CA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1636218-A1 THIAZOLYLPIPERIDINE DERIVATIVES AS MTP INHIBITORS MERCK PATENT GmbH (DE) 2006-03-22 EP disclosed
WO-2005003128-A1 THIAZOLYLPIPERIDINE DERIVATIVES AS MTP INHIBITORS MERCK PATENT GMBH (DE) 2005-01-13 WO disclosed