SCHEMBL5801474

SCHEMBL5801474

c1cnn2c(-c3ccncc3)nnc2c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MKNK1 Q9BUB5 1/20 0.53
HPGD P15428 7/20 0.44
SMN1; SMN2 Q16637 3/20 0.44
APAF1 O14727 2/20 0.44
RECQL P46063 1/20 0.44
HSD17B10 Q99714 9/20 0.43
ALDH1A1 P00352 7/20 0.43
MAPK1 P28482 4/20 0.43
KDM4E B2RXH2 4/20 0.43
TSHR P16473 2/20 0.43
TDP1 Q9NUW8 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
LRRK2 Q5S007 2/20 0.42
TP53 P04637 2/20 0.42
BRD4 O60885 1/20 0.41
ADORA3 P0DMS8 1/20 0.41
ADORA2A P29274 1/20 0.41
ADORA2B P29275 1/20 0.41
ADORA1 P30542 1/20 0.41
CREBBP Q92793 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2750732 0.87 BRD4 (0.54) HPGDSMN1; SMN2HSD17B10ALDH1A1MAPK1
SCHEMBL2804193 0.82 KDM4E (0.54) HPGDSMN1; SMN2HSD17B10ALDH1A1KDM4E
SCHEMBL22322759 0.81 MKNK1 (0.41) MKNK1HPGDSMN1; SMN2HSD17B10ALDH1A1
SCHEMBL4292173 0.75 LRRK2 (0.46) LRRK2
SCHEMBL12910190 0.73 KDM4E (0.55) HPGDSMN1; SMN2APAF1RECQLHSD17B10
SCHEMBL19957717 0.72 MKNK1 (0.42) MKNK1
SCHEMBL16417549 0.72 SMN1; SMN2 (0.41) MKNK1HPGDSMN1; SMN2HSD17B10ALDH1A1
SCHEMBL23458576 0.70 KDM4E (0.67) HPGDSMN1; SMN2APAF1RECQLHSD17B10
SCHEMBL1042919 0.70 DCTPP1 (0.44) ALDH1A1KDM4E
SCHEMBL1744648 0.69 MKNK1 (1.00) MKNK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021110890-A1 PYRIDINIUM DERIVATIVES AS HERBICIDES SYNGENTA CROP PROTECTION AG (CH) 2021-06-10 WO disclosed
WO-2021110890-A1 PYRIDINIUM DERIVATIVES AS HERBICIDES SYNGENTA CROP PROTECTION AG (CH) 2021-06-10 WO disclosed
EP-1691811-A1 COMBINATION OF A SEDATIVE AND A NEUROTRANSMITTER MODULATOR, AND METHODS FOR IMPROVING SLEEP QUALITY AND TREATING DEPRESSION Sepracor, Inc. (US) 2006-08-23 EP disclosed
WO-2005060968-A1 COMBINATION OF A SEDATIVE AND A NEUROTRANSMITTER MODULATOR, AND METHODS FOR IMPROVING SLEEP QUALITY AND TREATING DEPRESSION SEPRACOR INC. (US) 2005-07-07 WO disclosed