SCHEMBL5801912

SCHEMBL5801912

COc1ccccc1-n1cc(C#N)cn1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTOR P42345 1/20 0.43
SLC2A1 P11166 2/20 0.42
SLC2A3 P11169 2/20 0.42
MGLL Q99685 1/20 0.41
HPGDS O60760 1/20 0.41
CREBBP Q92793 2/20 0.41
DRD2 P14416 5/20 0.41
DRD3 P35462 4/20 0.41
DRD4 P21917 2/20 0.41
HTR1A P08908 1/20 0.41
HTR3E A5X5Y0 1/20 0.40
HTR3B O95264 1/20 0.40
ADRB1 P08588 1/20 0.40
CYP2C19 P33261 1/20 0.40
HTR3A P46098 1/20 0.40
HTR6 P50406 1/20 0.40
HTR3D Q70Z44 1/20 0.40
HTR3C Q8WXA8 1/20 0.40
SIGMAR1 Q99720 1/20 0.40
NPC1 O15118 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14330835 0.78 MTOR (0.46) MTORMGLLDRD2DRD3DRD4
SCHEMBL30239650 0.76 GRM4 (0.45) MTORMGLLDRD2DRD3DRD4
SCHEMBL21877535 0.76 DRD2 (0.46) MTORSLC2A1SLC2A3MGLLDRD2
SCHEMBL27686519 0.76 BCHE (0.41) MTORMGLLDRD2DRD3DRD4
SCHEMBL31297077 0.76 DRD2 (0.46) MTORSLC2A1SLC2A3MGLLDRD2
SCHEMBL23403311 0.76 GAA (0.51) MTORMGLLDRD2DRD3DRD4
SCHEMBL5804713 0.76 GRM4 (0.45) MTORMGLLDRD2DRD3DRD4
SCHEMBL22633031 0.76 MTOR (0.45) MTORMGLLDRD2DRD3DRD4
SCHEMBL30632073 0.76 GAA (0.51) MTORMGLLDRD2DRD3DRD4
SCHEMBL7805608 0.75 AVPR2 (0.49) MTORMGLLCREBBPDRD2DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1628980-A1 6-ARYLMETHYL-SUBSTITUTED PYRAZOLOPYRIMIDINES Bayer HealthCare AG (DE) 2006-03-01 EP disclosed
EP-1626971-A1 6-CYCLYLMETHYL- AND 6-ALKYLMETHYL-SUBSTITUTED PYRAZOLOPYRIMIDINES Bayer HealthCare AG (DE) 2006-02-22 EP disclosed
WO-2004099211-A1 6-CYCLYLMETHYL- AND 6-ALKYLMETHYL-SUBSTITUTED PYRAZOLOPYRIMIDINES BAYER HEALTHCARE AG (DE) 2004-11-18 WO disclosed
WO-2004099210-A1 6-ARYLMETHYL-SUBSTITUTED PYRAZOLOPYRIMIDINES BAYER HEALTHCARE AG (DE) 2004-11-18 WO disclosed