SCHEMBL5804378

SCHEMBL5804378

CCCCCC1(C)SC(=O)NC1=O

nearest known ligand 0.50

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.50
HSD11B1 P28845 11/20 0.43
CPT1A P50416 1/20 0.43
MMP2 P08253 3/20 0.36
MMP9 P14780 3/20 0.36
MMP3 P08254 1/20 0.36
MMP8 P22894 2/20 0.35
MMP13 P45452 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14209447 0.77 ALDH1A1 (0.59) ALDH1A1HSD11B1
SCHEMBL4202184 0.68 CPT1A (0.60) CPT1AMMP2MMP9MMP3MMP8
SCHEMBL13946478 0.68 CPT1A (0.60) CPT1AMMP2MMP9MMP3MMP8
SCHEMBL4209051 0.68 CPT1A (0.60) CPT1AMMP2MMP9MMP3MMP8
SCHEMBL13946474 0.68 CPT1A (0.60) CPT1AMMP2MMP9MMP3MMP8
SCHEMBL4204181 0.68 CPT1A (0.60) CPT1AMMP2MMP9MMP3MMP8
SCHEMBL11162084 0.67 CPT1A (0.41) CPT1A
SCHEMBL15413177 0.67 ALDH1A1 (1.00) ALDH1A1HSD11B1
SCHEMBL13547584 0.66 CPT1A (0.43) ALDH1A1CPT1AMMP2MMP9MMP3
SCHEMBL13332268 0.66 CPT1A (0.43) CPT1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1194146-B1 ARYLTHIAZOLIDINEDIONE AND ARYLOXAZOLIDINEDIONE DERIVATIVES MERCK & CO INC (US) 2006-07-19 EP disclosed
EP-1673059-A2 ALKANOL AND CYCLOALKANOL-AMINE DERIVATIVES AND METHODS OF THEIR USE Wyeth (US) 2006-06-28 EP disclosed
WO-2005037207-A2 ARYLALKYL-PIPERAZINE DERIVATIVES FOR THE TREATMENT OF CONDITIONS AMELIORATED BY MONOAMINE REUPTAKE INCLUDING VASOMOTOR SYMPTOMS (VMS) WYETH (US) 2005-04-28 WO disclosed
EP-1194146-A4 ARYLTHIAZOLIDINEDIONE AND ARYLOXAZOLIDINEDIONE DERIVATIVES MERCK & CO INC (US) 2002-07-31 EP disclosed
US-6399640-B1 ANTIDIABETIC AGENTS; ANTICHOLESTEROL AGENTS MERCK & CO., INC. 2002-06-04 US disclosed
EP-1194146-A1 ARYLTHIAZOLIDINEDIONE AND ARYLOXAZOLIDINEDIONE DERIVATIVES Merck & Co., Inc. (US) 2002-04-10 EP disclosed
WO-2000078312-A1 ARYLTHIAZOLIDINEDIONE AND ARYLOXAZOLIDINEDIONE DERIVATIVES MERCK & CO., INC. (US) 2000-12-28 WO disclosed